SCHEMBL21795640

SCHEMBL21795640

CC(=O)c1ccc(OCC2COCCC2OC(N)=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP15 Q460N3 4/20 0.42
PARP10 Q53GL7 4/20 0.42
PARP2 Q9UGN5 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
GAA P10253 2/20 0.40
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPT P10636 2/20 0.39
HRH2 P25021 1/20 0.38
HRH1 P35367 1/20 0.38
POLB P06746 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAOB P27338 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL15420637 0.82 PARP15 (0.45) PARP15PARP10PARP2L3MBTL1ALDH1A1
SCHEMBL21795659 0.81 NPC1 (0.39) PARP15PARP10PARP2SMN1; SMN2MAPT
SCHEMBL21795643 0.78 DDB1 (0.38) LMNA
SCHEMBL21795663 0.77 XDH (0.39)
SCHEMBL21795648 0.77 XDH (0.39) MAOB
SCHEMBL21795636 0.77 XDH (0.39) MAOB
SCHEMBL15420332 0.77 ALDH1A1 (0.42) L3MBTL1ALDH1A1KDM4EGAALMNA
SCHEMBL21795638 0.76 KDM4E (0.42) PARP2L3MBTL1ALDH1A1KDM4E
SCHEMBL21795642 0.76 GCG (0.34) PARP2ALDH1A1
SCHEMBL21795658 0.75 HDAC1 (0.39) KDM4EGAASMN1; SMN2MAPTMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2694472-B1 SULFONAMIDE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2020-03-11 EP disclosed