SCHEMBL2182545

SCHEMBL2182545

CC(=O)Oc1ccc(C2=Cc3ccc(OC(C)=O)cc3OC2c2cccnc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.46
TP53 P04637 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
PKM P14618 1/20 0.46
KMT2A Q03164 6/20 0.39
NFKB1 P19838 2/20 0.37
NFKB2 Q00653 2/20 0.37
RELA Q04206 2/20 0.37
CYP19A1 P11511 1/20 0.37
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
CA2 P00918 1/20 0.36
CA5A P35218 1/20 0.36
LMNA P02545 2/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12413304 0.93 RAB9A (0.44) NPC1TP53RAB9ASMN1; SMN2PKM
SCHEMBL2183468 0.87 NFKB1 (0.42) NPC1TP53RAB9ASMN1; SMN2PKM
SCHEMBL2181830 0.87 LMNA (0.42) NPC1KMT2ANFKB1NFKB2RELA
SCHEMBL12413324 0.80 ESR1 (0.39) NPC1TP53RAB9ASMN1; SMN2PKM
SCHEMBL12413374 0.80 LMNA (0.40) KMT2ANFKB1NFKB2RELAESR1
SCHEMBL12503744 0.78 RAB9A (0.40) NPC1TP53RAB9ASMN1; SMN2PKM
SCHEMBL2182453 0.78 ESR1 (0.48) CYP19A1ESR1ESR2LMNACYP11B1
SCHEMBL2182312 0.77 CA2 (0.44) TP53RAB9ASMN1; SMN2PKMKMT2A
SCHEMBL2180009 0.77 CA2 (0.44) TP53RAB9ASMN1; SMN2PKMKMT2A
SCHEMBL12503753 0.76 CA2 (0.37) NPC1TP53RAB9ASMN1; SMN2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110166142-A1 2-SUBSTITUTED ISOFLAVONOID COMPOUNDS, MEDICAMENTS AND USES NOVOGEN RESEARCH PTY LIMITED (AU) 2011-07-07 US disclosed
US-20110166142-A1 2-SUBSTITUTED ISOFLAVONOID COMPOUNDS, MEDICAMENTS AND USES NOVOGEN RESEARCH PTY LIMITED (AU) 2011-07-07 US disclosed
WO-2009003229-A1 2-SUBSTITUTED ISOFLAVONOID COMPOUNDS, MEDICAMENTS AND USES NOVOGEN RESEARCH PTY LTD (AU) 2009-01-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166142-A1 2-SUBSTITUTED ISOFLAVONOID COMPOUNDS, MEDICAMENTS AND USES NFE2L2, PTGS2, PTGES2 NPC1 1314/4885TP53 2490/4885RAB9A 4671/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.