SCHEMBL2186997

SCHEMBL2186997

NC(=Nc1nc2ccccc2[nH]1)NC(=O)c1csc(NC(=O)c2ccc(F)c(F)c2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.41
NPC1 O15118 8/20 0.39
RAB9A P51151 8/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
TP53 P04637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAOB P27338 1/20 0.39
MTOR P42345 1/20 0.38
CSNK1E P49674 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
MAPKAPK2 P49137 3/20 0.37
MAPK1 P28482 2/20 0.37
MAP2K1 Q02750 2/20 0.37
GAA P10253 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CSNK1D P48730 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2186602 0.91 FOXO1 (0.40) IRAK4NPC1RAB9ASMN1; SMN2TP53
SCHEMBL2187052 0.90 NPC1 (0.50) NPC1RAB9ASMN1; SMN2TP53KDM4E
SCHEMBL2187178 0.87 CSNK1D (0.45) NPC1RAB9ASMN1; SMN2TP53KDM4E
SCHEMBL2186693 0.87 MMP2 (0.46) NPC1RAB9ASMN1; SMN2TP53KDM4E
SCHEMBL2186979 0.87 MAPT (0.44) NPC1RAB9ASMN1; SMN2TP53KDM4E
SCHEMBL2189024 0.83 CSNK1E (0.49) NPC1SMN1; SMN2TP53PKMMTOR
SCHEMBL2186995 0.81 IRAK4 (0.51) IRAK4NPC1RAB9ASMN1; SMN2TP53
SCHEMBL2187310 0.79 NPC1 (0.52) NPC1RAB9ASMN1; SMN2KDM4EPKM
SCHEMBL2189072 0.79 CSNK1E (0.58) NPC1RAB9ATP53PKMMTOR
SCHEMBL2185628 0.77 SMN1; SMN2 (0.39) NPC1RAB9ASMN1; SMN2CSNK1EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343293-A1 NOVEL PIPERIDIN-4-YL-THIAZOLE-CARBOXAMIDE ANALOGUES AS INHIBITORS OF T-CELL PROLIFERATION AND USES THEREOF 4SC AG (DE) 2011-07-13 EP disclosed