SCHEMBL2187686

SCHEMBL2187686

NC(=NC(=O)c1csc(N2CCOCC2)n1)Nc1nc2ccccc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
MAPK1 P28482 2/20 0.46
GAA P10253 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
MAPT P10636 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
CYP3A4 P08684 1/20 0.45
KDM4E B2RXH2 1/20 0.43
CASR P41180 1/20 0.43
LMNA P02545 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2187578 0.85 TDP1 (0.46) SMN1; SMN2NPC1RAB9AMAPK1GAA
SCHEMBL2187668 0.81 KMT2A (0.48) SMN1; SMN2NPC1RAB9AMAPK1GAA
SCHEMBL2187530 0.75 SMN1; SMN2 (0.47) SMN1; SMN2NPC1RAB9ATDP1CYP3A4
SCHEMBL2186531 0.72 NFKB1 (0.41) SMN1; SMN2NPC1RAB9AGAATDP1
SCHEMBL2187394 0.71 IRAK4 (0.49) L3MBTL1
Hydrochloric Acid SCHEMBL5008548 0.68 L3MBTL1 (0.54) SMN1; SMN2NPC1RAB9ALMNAL3MBTL1
SCHEMBL16767096 0.68 CSNK1E (0.53) L3MBTL1
SCHEMBL18619678 0.67 LMNA (0.55) LMNAL3MBTL1
SCHEMBL2187574 0.67 GAA (0.44) SMN1; SMN2NPC1RAB9AMAPK1GAA
SCHEMBL420357 0.65 AR (0.54) SMN1; SMN2NPC1RAB9ALMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343293-A1 NOVEL PIPERIDIN-4-YL-THIAZOLE-CARBOXAMIDE ANALOGUES AS INHIBITORS OF T-CELL PROLIFERATION AND USES THEREOF 4SC AG (DE) 2011-07-13 EP disclosed