SCHEMBL2188126

SCHEMBL2188126

O=C(Cc1ccccc1)N1CCC(c2nc(C(=O)N3CCC(c4c[nH]c5ccccc45)CC3)cs2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 1/20 0.50
BRD4 O60885 1/20 0.50
POLB P06746 1/20 0.50
CREBBP Q92793 1/20 0.50
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CHRM4 P08173 1/20 0.46
SPR P35270 7/20 0.45
HSD11B1 P28845 1/20 0.44
TACR1 P25103 1/20 0.44
TACR3 P29371 1/20 0.44
ACACB O00763 1/20 0.44
ACACA Q13085 1/20 0.44
CCR2 P41597 2/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2186733 0.88 KDM4E (0.48) ALDH1A1KDM4EBRD4POLBCREBBP
SCHEMBL2188470 0.83 KDM4E (0.51) ALDH1A1KDM4EBRD4POLBCREBBP
SCHEMBL2213735 0.82 KDM4E (0.52) ALDH1A1KDM4EBRD4POLBCREBBP
SCHEMBL5774732 0.81 KDM4E (0.43) ALDH1A1KDM4EBRD4POLBCREBBP
SCHEMBL5287621 0.81 TACR1 (0.54) ALDH1A1KDM4EBRD4POLBCREBBP
SCHEMBL2186025 0.80 KDM4E (0.46) ALDH1A1KDM4EBRD4POLBCREBBP
SCHEMBL5769877 0.80 NPSR1 (0.51) ALDH1A1KDM4EPOLBLMNAHTT
SCHEMBL27698607 0.78 KMT2A (0.46) ALDH1A1KDM4EBRD4POLBCREBBP
SCHEMBL27698609 0.78 KMT2A (0.45) ALDH1A1KDM4EBRD4POLBCREBBP
SCHEMBL2187329 0.78 SLC6A4 (0.45) ALDH1A1KDM4EBRD4POLBCREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343293-A1 NOVEL PIPERIDIN-4-YL-THIAZOLE-CARBOXAMIDE ANALOGUES AS INHIBITORS OF T-CELL PROLIFERATION AND USES THEREOF 4SC AG (DE) 2011-07-13 EP disclosed
EP-1637529-A1 Novel piperidin-4-yl-thiazole-carboxamide analogues as inhibitors of T-cell proliferation and uses thereof 4SC AG (DE) 2006-03-22 EP disclosed