SCHEMBL27698609

SCHEMBL27698609

O=CC(CN1CCC(c2nc(C(=O)N3CCC(c4c[nH]c5ccccc45)CC3)cs2)CC1)c1ccc(F)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.45
KDM4E B2RXH2 1/20 0.43
BRD4 O60885 1/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
CREBBP Q92793 1/20 0.43
CCR2 P41597 7/20 0.42
SPR P35270 4/20 0.41
CHRM4 P08173 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRK1 P41145 1/20 0.39
OPRL1 P41146 1/20 0.39
HTR2A P28223 3/20 0.39
HTR7 P34969 3/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27698607 0.90 KMT2A (0.46) KMT2AKDM4EBRD4ALDH1A1POLB
SCHEMBL2186025 0.85 KDM4E (0.46) KMT2AKDM4EBRD4ALDH1A1POLB
SCHEMBL2186733 0.80 KDM4E (0.48) KMT2AKDM4EBRD4ALDH1A1POLB
SCHEMBL2188126 0.78 ALDH1A1 (0.50) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL2188470 0.77 KDM4E (0.51) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL2213735 0.75 KDM4E (0.52) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL5774731 0.73 CCR2 (0.41) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL5774732 0.72 KDM4E (0.43) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL2185602 0.70 KDM4E (0.45) KDM4EBRD4ALDH1A1POLBCREBBP
SCHEMBL2187684 0.70 HSD11B1 (0.48) KDM4EBRD4ALDH1A1POLBCREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101031567-B Novel heterocyclic NF-kB inhibitors 4SC Corp.,Ltd. (DE) 2011-12-21 CN claimed
CN-101031567-B Novel heterocyclic NF-kB inhibitors 4SC Corp.,Ltd. (DE) 2011-12-21 CN disclosed
CN-101031567-A Novel heterocyclic NF-kB inhibitors 4SC AG (DE) 2007-09-05 CN disclosed