SCHEMBL21883559

SCHEMBL21883559

CCCCCCc1cc(F)cc(C(N)=O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 2/20 0.46
PTGS2 P35354 3/20 0.46
TRPV1 Q8NER1 1/20 0.44
PLK1 P53350 1/20 0.43
PLK3 Q9H4B4 1/20 0.43
THRA P10827 4/20 0.43
THRB P10828 4/20 0.43
CYP3A4 P08684 1/20 0.43
RARB P10826 7/20 0.43
RARA P10276 2/20 0.43
RARG P13631 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
APAF1 O14727 1/20 0.42
RGS12 O14924 1/20 0.42
HSP90AA1 P07900 1/20 0.42
MAPK1 P28482 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
MTOR P42345 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9970966 0.80 PARP1 (0.46) PTGS2MEN1KMT2AALDH1A1
SCHEMBL15780156 0.78 GPR84 (0.58) GPR84PTGS2THRATHRBCYP3A4
SCHEMBL9243315 0.77 PTGS2 (0.56) GPR84PTGS2TRPV1CYP3A4MAPK1
SCHEMBL15964806 0.76 SPHK2 (0.60)
SCHEMBL28241905 0.76 SPHK2 (0.60)
SCHEMBL9356792 0.76 SPHK2 (0.60)
SCHEMBL201440 0.76 PLA2G2A (0.59) CYP3A4RARBMEN1KMT2AMAPT
SCHEMBL6835676 0.75 THRA (0.65) THRATHRBRARBRARAMEN1
SCHEMBL13617729 0.75 THRA (0.65) THRATHRBRARBRARAMEN1
SCHEMBL351935 0.75 THRA (0.65) THRATHRBRARBRARAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10597377-B2 Somatostatin modulators and uses thereof Crinetics Pharmaceuticals, Inc. (US) 2020-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10597377-B2 Somatostatin modulators and uses thereof SSTR5, SSTR2, SSTR4 GPR84 365/4885PTGS2 1938/4885TRPV1 894/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.