SCHEMBL2188442

SCHEMBL2188442

O=C(Cc1ccc(F)cc1)N1CCC(c2nc(C(=O)N3CCc4ccccc4C3)cs2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.47
RAB9A P51151 3/20 0.47
PDE4B Q07343 2/20 0.45
PDE4D Q08499 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
LMNA P02545 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
TRPC3 Q13507 2/20 0.43
TRPC6 Q9Y210 2/20 0.43
MDM2 Q00987 1/20 0.43
GAA P10253 1/20 0.41
ROCK2 O75116 1/20 0.41
ALDH1A1 P00352 2/20 0.40
CNR1 P21554 1/20 0.40
PKM P14618 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2188486 0.90 MAPK1 (0.40) NPC1RAB9AKMT2ALMNAALOX15
SCHEMBL2186946 0.87 LMNA (0.46) NPC1RAB9ALMNAALOX15TSHR
SCHEMBL2186625 0.83 MAPT (0.56) RAB9AMEN1KMT2ALMNAALOX15
SCHEMBL27679675 0.82 LMNA (0.50) MEN1KMT2ALMNAALOX15TSHR
SCHEMBL2185718 0.81 LMNA (0.40) RAB9ALMNAALOX15TSHRMAPK1
SCHEMBL2188722 0.81 KDM4E (0.57) NPC1RAB9AMEN1KMT2ALMNA
SCHEMBL2186974 0.81 CACNA2D1 (0.48) NPC1RAB9AMEN1KMT2ALMNA
SCHEMBL2186813 0.79 SCD5 (0.43) LMNAALOX15TSHRMAPK1TRPC3
SCHEMBL2188684 0.79 KMT2A (0.39) KMT2ALMNAALOX15TSHRMAPK1
SCHEMBL2187333 0.79 MAPT (0.51) KMT2ALMNAALOX15TSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343293-A1 NOVEL PIPERIDIN-4-YL-THIAZOLE-CARBOXAMIDE ANALOGUES AS INHIBITORS OF T-CELL PROLIFERATION AND USES THEREOF 4SC AG (DE) 2011-07-13 EP disclosed