SCHEMBL21929341

SCHEMBL21929341

COc1cccc(COC2=CC(=O)N[C@H]2Cc2ccccc2)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOB P27338 7/20 0.48
HTR1A P08908 3/20 0.43
ABCB1 P08183 2/20 0.43
DRD2 P14416 2/20 0.43
MRGPRX4 Q96LA9 1/20 0.43
IDO1 P14902 2/20 0.43
AGXT P21549 2/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
MMP1 P03956 1/20 0.42
MMP3 P08254 1/20 0.42
MMP9 P14780 1/20 0.42
MAOA P21397 1/20 0.42
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
KDM1A O60341 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20734910 0.88 MMP1 (0.48) MAOBABCB1NPC1RAB9AMMP1
SCHEMBL20734898 0.84 TSHR (0.45) ABCB1IDO1MMP1MMP3MMP9
SCHEMBL20734899 0.84 TSHR (0.45) ABCB1IDO1MMP1MMP3MMP9
SCHEMBL20734912 0.83 ALOX5 (0.42) MAOBMRGPRX4RAB9AMAOA
SCHEMBL20734901 0.83 P2RX7 (0.46) MAOBIDO1AGXTMAOA
SCHEMBL20734907 0.83 ALOX5 (0.42) MAOBMRGPRX4RAB9AMAOA
SCHEMBL20734900 0.83 P2RX7 (0.46) MAOBIDO1AGXTMAOA
SCHEMBL20734807 0.80 ALDH1A1 (0.44) NPC1RAB9A
SCHEMBL20734808 0.80 ALDH1A1 (0.44) NPC1RAB9A
SCHEMBL20734921 0.79 HRH3 (0.47) MMP1MMP3MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3643311-A1 4-OXO-ALKYLATED TETRAMIC ACID COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF Beijing Joekai Biotech. LLC (CN) 2020-04-29 EP disclosed