SCHEMBL21938565

SCHEMBL21938565

CCCc1cc2cn[nH]c2cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 4/20 0.50
ROCK2 O75116 4/20 0.50
GSK3B P49841 3/20 0.50
JAK2 O60674 2/20 0.50
ROCK1 Q13464 2/20 0.50
AURKB Q96GD4 2/20 0.50
AURKA O14965 1/20 0.50
DAPK3 O43293 1/20 0.50
CHEK2 O96017 1/20 0.50
CDK2 P24941 1/20 0.50
MARK3 P27448 1/20 0.50
GSK3A P49840 1/20 0.50
LIMK1 P53667 1/20 0.50
CDK5 Q00535 1/20 0.50
DYRK1A Q13627 1/20 0.50
PRKD2 Q9BZL6 1/20 0.50
CHEK1 O14757 1/20 0.40
AXL P30530 1/20 0.40
MKNK1 Q9BUB5 4/20 0.40
PIM3 Q86V86 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10235446 0.85 TRPA1 (0.43) PIM1ROCK2GSK3BJAK2ROCK1
SCHEMBL13940969 0.78 CHEK1 (0.47) PIM1ROCK2GSK3BROCK1CDK2
SCHEMBL15541878 0.78 CHEK1 (0.42) PIM1ROCK2GSK3BROCK1CDK2
SCHEMBL4996798 0.78 DYRK1A (0.48) PIM1ROCK2GSK3BJAK2ROCK1
SCHEMBL25107119 0.78 PIM1 (0.39) PIM1ROCK2GSK3BJAK2ROCK1
SCHEMBL20627222 0.77 CHEK1 (0.39) PIM1ROCK2GSK3BJAK2ROCK1
SCHEMBL23119370 0.77 NOS1 (0.41) PIM1ROCK2GSK3BJAK2ROCK1
Hydrochloric Acid SCHEMBL7221088 0.76 CHEK1 (0.46) PIM1ROCK2GSK3BROCK1CDK2
SCHEMBL24493489 0.74 GABRP (0.41) GABRPGABRDGABRA1IDO1GABRB1
SCHEMBL8220180 0.71 ROCK2 (0.54) PIM1ROCK2GSK3BJAK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2986624-B1 19-NOR NEUROACTIVE STEROIDS FOR METHODS OF TREATMENT SAGE THERAPEUTICS INC (US) 2020-03-25 EP disclosed