SCHEMBL21964572

SCHEMBL21964572

CNC(O)c1cc([N+](=O)[O-])nn1C1CCCC1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CMKLR1 Q99788 2/20 0.33
POLB P06746 1/20 0.33
PTGS2 P35354 2/20 0.33
MAPK13 O15264 1/20 0.32
MAPK12 P53778 1/20 0.32
MAPK11 Q15759 1/20 0.32
MAPK14 Q16539 1/20 0.32
HTT P42858 1/20 0.32
PDE7A Q13946 1/20 0.31
KCNJ6 P48051 1/20 0.31
KCNJ5 P48544 1/20 0.31
KCNJ3 P48549 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HCAR3 P49019 2/20 0.30
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
KMT2A Q03164 1/20 0.30
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2373603 0.75 HCAR3 (0.38) POLBPTGS2MAPK13MAPK12MAPK11
SCHEMBL21960367 0.74 OPRK1 (0.39) POLBPTGS2PDE7AALDH1A1MEN1
SCHEMBL15767938 0.72 POLB (0.34) CMKLR1POLBPTGS2MAPK13MAPK12
SCHEMBL21960888 0.68 BAZ2B (0.39) POLBPDE7AALDH1A1MEN1KMT2A
SCHEMBL21960936 0.68 PKM (0.40) POLBALDH1A1MEN1KMT2A
SCHEMBL21961446 0.68 PTGS2 (0.41) PTGS2
SCHEMBL25405989 0.62 CYP4F2 (0.41) POLBHTTALDH1A1MEN1KMT2A
SCHEMBL31018603 0.62 F2 (0.40) HTTKCNJ6KCNJ5KCNJ3ALDH1A1
SCHEMBL31052556 0.61 MAPT (0.47) KCNJ6KCNJ5KCNJ3ALDH1A1MEN1
SCHEMBL2053383 0.60 ALDH1A1 (0.34) POLBALDH1A1HCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3478675-B1 HETEROAROMATIC DERIVATIVES AS NIK INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2020-04-22 EP disclosed