SCHEMBL2198935

SCHEMBL2198935

CC(=O)c1ccc(Cl)c(S(=O)(=O)Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.46
KMT2A Q03164 2/20 0.46
TP53 P04637 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
CYP1A2 P05177 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
POLB P06746 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CA1 P00915 4/20 0.42
CA2 P00918 4/20 0.42
MEN1 O00255 1/20 0.41
NPBWR1 P48145 1/20 0.41
MCHR1 Q99705 1/20 0.41
ATAD2 Q6PL18 1/20 0.40
CECR2 Q9BXF3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1495711 0.85 SMN1; SMN2 (0.46) SMN1; SMN2KMT2ATP53TDP1ALDH1A1
SCHEMBL7143525 0.84 CA1 (0.58) HSD17B10CA1CA2
SCHEMBL396004 0.83 TDP1 (0.61) SMN1; SMN2KMT2ATDP1ALDH1A1L3MBTL1
SCHEMBL1926208 0.83 TDP1 (0.45) SMN1; SMN2KMT2ATDP1ALDH1A1L3MBTL1
SCHEMBL10652398 0.81 PKM (0.49) SMN1; SMN2ALDH1A1POLBCA1CA2
SCHEMBL9548071 0.81 PTGER4 (0.45) SMN1; SMN2TDP1L3MBTL1POLB
SCHEMBL1925386 0.81 SMN1; SMN2 (0.47) SMN1; SMN2KMT2ATDP1ALDH1A1L3MBTL1
SCHEMBL21183474 0.81 POLB (0.50) SMN1; SMN2KMT2ATP53TDP1ALDH1A1
SCHEMBL11595745 0.81 GSTO1 (0.57) SMN1; SMN2KMT2AALDH1A1L3MBTL1CYP1A2
SCHEMBL1495720 0.81 ALDH1A1 (0.65) SMN1; SMN2KMT2ATDP1ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11912668-B2 GCN2 and perk kinase inhibitors and methods of use thereof DECIPHERA PHARMACEUTICALS, LLC (US) 2024-02-27 US disclosed
US-11912668-B2 GCN2 and perk kinase inhibitors and methods of use thereof DECIPHERA PHARMACEUTICALS, LLC (US) 2024-02-27 US disclosed
WO-2022109001-A1 GCN2 AND PERK KINASE INHIBITORS AND METHODS OF USE THEREOF DECIPHERA PHARMACEUTICALS, LLC (US) 2022-05-27 WO disclosed
EP-1658263-B9 NOVEL AMINOBENZOPHENONE COMPOUNDS LEO PHARMA AS (DK) 2011-11-09 EP disclosed
US-7977387-B2 Aminobenzophenone compounds LEO PHARMA A/S (DK) 2011-07-12 US disclosed
EP-1658263-B1 NOVEL AMINOBENZOPHENONE COMPOUNDS LEO PHARMA AS (DK) 2010-06-02 EP disclosed
US-20060166990-A1 Novel aminobenzophenone compounds LEO PHARMA A/S (DK) 2006-07-27 US disclosed
EP-1658263-A1 NOVEL AMINOBENZOPHENONE COMPOUNDS Leo Pharma A/S (DK) 2006-05-24 EP disclosed
WO-2005009940-A1 NOVEL AMINOBENZOPHENONE COMPOUNDS LEO PHARMA A/S (DK) 2005-02-03 WO disclosed
US-4125614-A DIURETIC HOECHST AKTIENGESELLSCHAFT (DE) 1978-11-14 US disclosed
US-4061761-A Thiazolidine derivatives HOECHST AKTIENGESELLSCHAFT (DT) 1977-12-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060166990-A1 Novel aminobenzophenone compounds NFKBIA, UACA, ALDH7A1 SMN1; SMN2 4625/4885KMT2A 3430/4885TP53 189/4885
US-11912668-B2 GCN2 and perk kinase inhibitors and methods of use thereof EIF2AK4, GCN1, MAPKAPK2 SMN1; SMN2 538/4885KMT2A 4116/4885TP53 3755/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.