SCHEMBL22014433

SCHEMBL22014433

CNCc1ccc(/[SH](=O)=N/C(=O)Cc2c(-c3ccccc3)ccc3c2CCC3)cc1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RXRA P19793 3/20 0.34
RXRB P28702 3/20 0.34
RXRG P48443 3/20 0.34
HDAC6 Q9UBN7 2/20 0.31
F7 P08709 3/20 0.31
METAP2 P50579 2/20 0.31
NQO1 P15559 2/20 0.31
F3 P13726 1/20 0.31
F2 P00734 1/20 0.30
ADRA1B P35368 1/20 0.30
LMNA P02545 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
TSHR P16473 1/20 0.30
AGTR2 P50052 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21962236 0.80 KMT2A (0.39) RXRARXRBRXRGMETAP2KMT2A
SCHEMBL25067101 0.80 KMT2A (0.39) RXRARXRBRXRGMETAP2KMT2A
SCHEMBL21962077 0.72 RXRB (0.43) RXRARXRBRXRGMETAP2LMNA
SCHEMBL22014435 0.70 POLB (0.36) RXRARXRBRXRGMETAP2NQO1
SCHEMBL21962126 0.70 MEN1 (0.39) RXRARXRBRXRGMETAP2NQO1
SCHEMBL21962078 0.67 MTNR1A (0.45) RXRARXRBRXRGMETAP2TSHR
SCHEMBL25033972 0.60 NLRP3 (0.40)
SCHEMBL28153404 0.58 NOS1 (0.39) SMN1; SMN2
SCHEMBL21500405 0.58 PARP1 (0.44) TSHR
SCHEMBL23692355 0.57 ALDH1A1 (0.35) LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102574-A1 THE COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed