Oglemilast

Oglemilast

SCHEMBL220245

CS(=O)(=O)Nc1ccc2oc3c(OC(F)F)ccc(C(=O)Nc4c(Cl)cncc4Cl)c3c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PDE4APDE4BPDE4CPDE4D

The experimentally established mechanism targets of Oglemilast. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4D known ✓ Q08499 15/20 1.00
PDE4B known ✓ Q07343 17/20 0.64
PDE4A known ✓ P27815 14/20 0.64
PDE4C known ✓ Q08493 13/20 0.64
ABCB11 O95342 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oglemilast SCHEMBL29413215 1.00 PDE4D (1.00) PDE4DPDE4BPDE4APDE4CABCB11
Oglemilast SCHEMBL29369504 1.00 PDE4D (1.00) PDE4DPDE4BPDE4APDE4CABCB11
Oglemilast SCHEMBL4030019 0.99 PDE4D (0.98) PDE4DPDE4BPDE4APDE4CABCB11
Oglemilast SCHEMBL4030005 0.99 PDE4D (0.98) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL4035094 0.92 PDE4D (0.85) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL4027253 0.91 PDE4D (0.84) PDE4DPDE4BPDE4APDE4C
SCHEMBL4029909 0.90 PDE4D (0.81) PDE4DPDE4BPDE4APDE4C
SCHEMBL13777247 0.89 PDE4D (0.81) PDE4DPDE4BPDE4APDE4C
SCHEMBL4030622 0.89 PDE4D (0.80) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL4029693 0.88 PDE4D (0.79) PDE4DPDE4BPDE4APDE4CABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 699 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4565302-A1 DRY POWDER INHALER Chiesi Farmaceutici S.p.A. (IT) 2025-06-11 EP claimed
US-11903992-B2 Composition comprising lidocaine, l-carnosine and dexpanthenol CELLIX BIO PRIVATE LIMITED (IN) 2024-02-20 US claimed
US-20240042147-A1 DRY POWDER INHALER CHIESI FARMACEUTICI S.P.A. (IT) 2024-02-08 US claimed
WO-2024028388-A1 DRY POWDER INHALER CHIESI FARMACEUTICI S.P.A. (IT) 2024-02-08 WO claimed
US-11504332-B2 Phosphodiesterase-4 inhibitor combinations, methods of making, and methods of use thereof VK RESEARCH ASSOCIATES INC. (US) 2022-11-22 US claimed
US-20220304935-A1 PHOSPHODIESTERASE-4 INHIBITOR COMBINATIONS, METHODS OF MAKING, AND METHODS OF USE THEREOF VK Research Associates Inc 2022-09-29 US claimed
WO-2022190030-A1 A TOPICAL FORMULATION FOR THE TREATMENT OF SKIN DISEASES AVACA PHARMA PRIVATE LIMITED (IN) 2022-09-15 WO claimed
US-11439627-B2 Pharmaceutical composition for the treatment of autism Stalicla S.A. (CH) 2022-09-13 US claimed
WO-2022157587-A1 A COMPOSITION COMPRISING LIDOCAINE, L-CARNOSINE AND DEXPANTHENOL CELLIX BIO PRIVATE LIMITED (IN) 2022-07-28 WO claimed
US-20220233629-A1 COMPOSITION COMPRISING LIDOCAINE, L-CARNOSINE AND DEXPANTHENOL CELLIX BIO PRIVATE LIMITED (IN) 2022-07-28 US claimed
WO-2008005955-A2 SYNTHESIS OF HETEROCYCLIC COMPOUNDS FOREST LABORATORIES HOLDINGS LIMITED (BM) 2008-01-10 WO claimed
US-20080009632-A1 SYNTHESIS OF HETEROCYCLIC COMPOUNDS FOREST LABORATORIES HOLDINGS LIMITED (BM) 2008-01-10 US claimed
EP-1799632-A2 PROCESS FOR THE PREPARATION OF N-(3,5-DICHLOROPYRID-4-YL)-4-DIFLUOROMETHOXY-8-METHANESULFONAMIDO-DIBENZO[B,D]FURAN-1-CARBOXAMIDE Glenmark Pharmaceuticals S.A. (CH) 2007-06-27 EP claimed
US-7223789-B2 Heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them GLENMARK PHARMACEUTICALS S.A. (CH) 2007-05-29 US claimed
US-20070105855-A1 NOVEL HETEROCYCLIC COMPOUNDS USEFUL FOR THE TREATMENT OF INFLAMMATORY AND ALLERGIC DISORDERS: PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLENMARK PHARMACEUTICALS S.A. (CH) 2007-05-10 US claimed
US-20060135779-A1 Process for the preparation n-(3,5-dichloropyrid-4-yl)-4-difluoromethoxy-8-methane sulfonamido-dibenzo[b,d]furan-1-carboxamide GLENMARK PHARMACEUTICALS S.A. (CH) 2006-06-22 US claimed
WO-2006040652-A2 PROCESS FOR THE PREPARATION OF N-(3,5-DICHLOROPYRID-4-YL)-4DIFLUOROMETHOXY-8-METHANESULFONAMIDO-DIBENZO[B,D]FURAN-1-CARBOXAMIDE GLENMARK PHARMACEUTICALS S.A. (US) 2006-04-20 WO claimed
EP-1620429-A1 NOVEL HETEROCYCLIC COMPOUNDS USEFUL FOR THE TREATMENT OF INFLAMMATORY AND ALLERGIC DISORDERS: PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Glenmark Pharmaceuticals S.A. (CH) 2006-02-01 EP claimed
US-20050027129-A1 Novel heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them GLENMARK PHARMACEUTICALS, INC. USA 2005-02-03 US claimed
WO-2004089940-A1 NOVEL HETEROCYCLIC COMPOUNDS USEFUL FOR THE TREATMENT OF INFLAMMATORY AND ALLERGIC DISORDERS: PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLENMARK PHARMACEUTICALS S.A. (US) 2004-10-21 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060135779-A1 Process for the preparation n-(3,5-dichloropyrid-4-yl)-4-difluoromethoxy-8-methane sulfonamido-dibenzo[b,d]furan-1-carboxamide HCN4, REN, QDPR PDE4D 378/4885PDE4B 696/4885PDE4A 1242/4885
US-20050027129-A1 Novel heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them PDE4A, PDE4B, PDE12 PDE4D 4/4885PDE4B 2/4885PDE4A 1/4885
US-20080009632-A1 SYNTHESIS OF HETEROCYCLIC COMPOUNDS FDPS, DHPS, AADAC PDE4D 1209/4885PDE4B 1634/4885PDE4A 2332/4885
US-20070105855-A1 NOVEL HETEROCYCLIC COMPOUNDS USEFUL FOR THE TREATMENT OF INFLAMMATORY AND ALLERGIC DISORDERS: PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM PDE4A, PDE4B, PDE12 PDE4D 4/4885PDE4B 2/4885PDE4A 1/4885
US-11903992-B2 Composition comprising lidocaine, l-carnosine and dexpanthenol VNN1, LPL, HMGB1 PDE4D 1677/4885PDE4B 1894/4885PDE4A 1073/4885
US-20220233629-A1 COMPOSITION COMPRISING LIDOCAINE, L-CARNOSINE AND DEXPANTHENOL VNN1, LPL, HMGB1 PDE4D 1677/4885PDE4B 1894/4885PDE4A 1073/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.