SCHEMBL22061395

SCHEMBL22061395

C=CCc1nc2ccnc(C)c2[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.39
MAPT P10636 2/20 0.36
TP53 P04637 1/20 0.36
ALDH1A1 P00352 4/20 0.34
HPGD P15428 4/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
KDM4E B2RXH2 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 2/20 0.34
HSD17B10 Q99714 2/20 0.34
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
GABRA1 P14867 1/20 0.34
TSHR P16473 1/20 0.34
GABRB1 P18505 1/20 0.34
GABRG2 P18507 1/20 0.34
NFKB1 P19838 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3258411 0.76 ALDH1A1 (0.39) MAPTTP53ALDH1A1HPGDMEN1
SCHEMBL18576288 0.72 MAOA (0.42) MAOAMAPTALDH1A1HPGDMEN1
SCHEMBL2378021 0.72 MAPT (0.44) MAPTTP53ALDH1A1MEN1KMT2A
SCHEMBL2163313 0.71 MAPT (0.40) MAPTTP53ALDH1A1HPGDMEN1
SCHEMBL4633992 0.70 RET (0.34) MAPTTP53ALDH1A1HPGDMEN1
SCHEMBL10634839 0.70 ACHE (0.36) MAPTALDH1A1HPGDMEN1KMT2A
SCHEMBL28154129 0.70 LMNA (0.36) MAPTALDH1A1HPGDMEN1KMT2A
SCHEMBL9228130 0.70 ALDH1A1 (0.39) MAPTTP53ALDH1A1HPGDMEN1
SCHEMBL12778762 0.69 MAOA (0.40) MAOAMAPTALDH1A1HPGDMEN1
SCHEMBL22962312 0.67 KDM4E (0.41) MAOAMAPTALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3139919-B1 COMPOUNDS FOR TREATMENT OF CANCER ONCTERNAL THERAPEUTICS INC (US) 2020-06-03 EP disclosed