SCHEMBL22101707

SCHEMBL22101707

CCc1nc2c(F)cc(C)cn2c(=O)c1OCC(N)=O

nearest known ligand 0.32

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MAPK14 Q16539 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
ADORA2A P29274 2/20 0.31
ADORA2B P29275 2/20 0.31
ADORA1 P30542 2/20 0.31
DPP4 P27487 1/20 0.31
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.31
KDM4E B2RXH2 3/20 0.31
HPGD P15428 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.30
POLB P06746 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
PIK3CA P42336 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22101713 0.87 MAPT (0.34) ALDH1A1RXFP1MAPTLMNAKDM4E
SCHEMBL22393762 0.86 BTK (0.31) ALDH1A1L3MBTL1MAPT
SCHEMBL22101917 0.86 P2RX3 (0.31) ALDH1A1L3MBTL1DPP4
SCHEMBL22101706 0.84 HTR1A (0.32) L3MBTL1MAPK14RXFP1MAPTLMNA
SCHEMBL22101184 0.82 CRHR1 (0.31) ALDH1A1LMNASMN1; SMN2
SCHEMBL22101905 0.82 PDE2A (0.31) ALDH1A1L3MBTL1RXFP1MAPTKDM4E
SCHEMBL22101709 0.77 GRIN1 (0.32) ALDH1A1RXFP1LMNAKDM4EHPGD
SCHEMBL22393703 0.74 SYK (0.37) ALDH1A1KDM4E
SCHEMBL23099580 0.72 NPC1 (0.33) ALDH1A1RXFP1LMNAHPGDGAA
SCHEMBL22393702 0.70 HCAR2 (0.32) L3MBTL1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed