SCHEMBL22101905

SCHEMBL22101905

CCc1nc2c(F)cc(C)cn2c(=O)c1OCCOC

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.31
MET P08581 2/20 0.31
RXFP1 Q9HBX9 1/20 0.31
KCNJ5 P48544 1/20 0.30
KCNJ3 P48549 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
HSD17B10 Q99714 1/20 0.30
ATM Q13315 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22393702 0.88 HCAR2 (0.32) METCYP1A2CYP3A4TSHRHSD17B10
SCHEMBL22101706 0.88 HTR1A (0.32) RXFP1KCNJ5KCNJ3ATML3MBTL1
SCHEMBL22101184 0.87 CRHR1 (0.31) ALDH1A1
SCHEMBL22393761 0.85 MET (0.30) MET
SCHEMBL22101707 0.82 ALDH1A1 (0.32) RXFP1HSD17B10L3MBTL1KDM4EALDH1A1
SCHEMBL22101713 0.80 MAPT (0.34) RXFP1TSHRKDM4EALDH1A1MAPT
SCHEMBL22101709 0.79 GRIN1 (0.32) RXFP1TSHRHSD17B10KDM4EALDH1A1
SCHEMBL22101539 0.78 FFAR4 (0.35) PDE2AMETRXFP1CYP1A2CYP3A4
SCHEMBL22101906 0.77 KDM4E (0.43) RXFP1KDM4EALDH1A1MAPT
SCHEMBL22393755 0.73 P2RX7 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed