SCHEMBL221260

SCHEMBL221260

CC(C)N1CCC(N(CC(F)(F)F)S(=O)(=O)CCN2C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.46
ACHE P22303 2/20 0.40
NLRP3 Q96P20 1/20 0.39
DRD2 P14416 2/20 0.35
SLC6A2 P23975 1/20 0.34
HTR1A P08908 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
DRD3 P35462 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL219546 0.83 MAOB (0.51) MAOBACHENLRP3DRD2
SCHEMBL222398 0.78 MAOB (0.41) MAOBACHENLRP3DRD2SLC6A2
SCHEMBL222333 0.73 MAOB (0.52) MAOBACHEDRD2HTR1A
SCHEMBL4592502 0.71 MAOB (0.50) MAOBACHE
SCHEMBL4592504 0.70 MAOB (0.49) MAOBACHEDRD2
SCHEMBL4592501 0.69 MAOB (0.48) MAOBACHE
SCHEMBL3761385 0.66 MAOB (0.50) MAOBACHENLRP3
SCHEMBL18673359 0.65 SLC6A2 (0.45) SLC6A2
SCHEMBL3876433 0.65 HTR2A (0.36) DRD2SLC6A2HTR1A
SCHEMBL3963524 0.64 MAOB (1.00) MAOBDRD2HTR1ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088925-B2 low molecular weight factor Xa specific blood clotting inhibitors; less side effects; 5-Chloro-thiophene-2-carboxylic acid [2-(1-isopropyl-piperidin-4-ylsulfamoyl)-ethyl]-amide; thromboembolic diseases or restenosis; antithrombotic agents SANOFI-AVENTIS (FR) 2012-01-03 US disclosed