SCHEMBL222333

SCHEMBL222333

CC(C)N1CCC(NS(=O)(=O)CCN2C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.52
F10 P00742 1/20 0.49
ACHE P22303 1/20 0.43
HTR1A P08908 3/20 0.43
HTR7 P34969 3/20 0.43
DRD2 P14416 1/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM1A O60341 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4592502 0.84 MAOB (0.50) MAOBACHEALDH1A1
SCHEMBL221237 0.83 ACHE (0.42) ACHEDRD2ALDH1A1KDM1A
SCHEMBL4592504 0.83 MAOB (0.49) MAOBACHEDRD2ALDH1A1KDM1A
SCHEMBL219755 0.78 HTR1A (0.42) MAOBACHEHTR1AALDH1A1KDM1A
SCHEMBL219546 0.78 MAOB (0.51) MAOBACHEDRD2
SCHEMBL19739574 0.75 HPGD (0.56) ACHEHTR1AHTR7ALDH1A1
SCHEMBL4592501 0.75 MAOB (0.48) MAOBACHEALDH1A1
Taltrimide SCHEMBL347001 0.74 NPSR1 (0.48) MAOBALDH1A1
Taltrimide SCHEMBL29866257 0.74 NPSR1 (0.48) MAOBALDH1A1
SCHEMBL13102745 0.73 F10 (0.49) F10HTR1AHTR7DRD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088925-B2 low molecular weight factor Xa specific blood clotting inhibitors; less side effects; 5-Chloro-thiophene-2-carboxylic acid [2-(1-isopropyl-piperidin-4-ylsulfamoyl)-ethyl]-amide; thromboembolic diseases or restenosis; antithrombotic agents SANOFI-AVENTIS (FR) 2012-01-03 US disclosed