SCHEMBL222398

SCHEMBL222398

CC(C)N1CCC(N(Cc2nccs2)S(=O)(=O)CCN2C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.41
NLRP3 Q96P20 1/20 0.38
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
SLC6A2 P23975 1/20 0.34
HPGD P15428 2/20 0.34
ACHE P22303 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 1/20 0.34
DRD2 P14416 1/20 0.34
XIAP P98170 1/20 0.33
CYP1B1 Q16678 1/20 0.33
PKM P14618 1/20 0.33
HTR1A P08908 1/20 0.33
SCN1A P35498 1/20 0.32
SCN8A Q9UQD0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL222300 0.82 HDAC6 (0.34) SCN1ASCN8A
SCHEMBL221260 0.78 MAOB (0.46) MAOBNLRP3SLC6A2ACHEDRD2
SCHEMBL219546 0.77 MAOB (0.51) MAOBNLRP3HPGDACHEHSD17B10
SCHEMBL3876208 0.76 HRH3 (0.37) SCN8A
SCHEMBL219979 0.72 F10 (0.58) ALDH1A1HPGD
SCHEMBL3876204 0.71 F10 (0.42)
SCHEMBL222333 0.68 MAOB (0.52) MAOBALDH1A1ACHEDRD2HTR1A
SCHEMBL4592502 0.67 MAOB (0.50) MAOBALDH1A1ACHEPKM
SCHEMBL4592504 0.66 MAOB (0.49) MAOBALDH1A1HPGDACHEDRD2
SCHEMBL4592501 0.65 MAOB (0.48) MAOBALDH1A1GAAHPGDACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088925-B2 low molecular weight factor Xa specific blood clotting inhibitors; less side effects; 5-Chloro-thiophene-2-carboxylic acid [2-(1-isopropyl-piperidin-4-ylsulfamoyl)-ethyl]-amide; thromboembolic diseases or restenosis; antithrombotic agents SANOFI-AVENTIS (FR) 2012-01-03 US disclosed