SCHEMBL22129172

SCHEMBL22129172

COC(=O)c1ccc2nccc(OCC(F)F)c2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.48
HTT P42858 2/20 0.48
KDM4E B2RXH2 4/20 0.41
KDM6B O15054 1/20 0.41
KDM5C P41229 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KDM2A Q9Y2K7 1/20 0.41
KDM3A Q9Y4C1 1/20 0.41
MET P08581 3/20 0.41
MAPT P10636 2/20 0.41
GSK3B P49841 1/20 0.41
AXL P30530 1/20 0.40
JMJD6 Q6NYC1 1/20 0.40
CYP2C9 P11712 1/20 0.39
DYRK1A Q13627 1/20 0.39
PAX8 Q06710 1/20 0.39
IDO1 P14902 3/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22129173 0.86 IDO1 (0.40) HTTKDM4EKDM6BKDM5CKDM4C
SCHEMBL22149303 0.85 IDO1 (0.41) METMAPTGSK3BAXLIDO1
SCHEMBL6301162 0.84 ALOX15 (0.57) ALOX15HTTKDM4EKDM6BKDM5C
SCHEMBL22149069 0.80 MAPT (0.37) ALOX15HTTMETMAPTGSK3B
SCHEMBL22129178 0.80 JMJD6 (0.39) ALOX15METMAPTGSK3BJMJD6
SCHEMBL22149079 0.78 MET (0.36) KDM4EMETMAPTGSK3BAXL
SCHEMBL6298726 0.77 ALOX15 (0.56) ALOX15HTTKDM4EKDM6BKDM5C
SCHEMBL31734085 0.77 ALOX15 (0.56) ALOX15HTTKDM4EKDM6BKDM5C
SCHEMBL22129170 0.77 JMJD6 (0.36) MAPTGSK3BJMJD6IDO1CYP3A4
SCHEMBL2716634 0.76 LMNA (0.50) HTTMAPTCYP2C9CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111670182-A Quinoline derivatives, preparation method and application thereof 东莞市东阳光农药研发有限公司 2020-09-15 CN disclosed
WO-2020124515-A1 QUINOLINE DERIVATIVE, PREPARATION METHOD AND USE THEREOF 东莞市东阳光农药研发有限公司 2020-06-25 WO disclosed
WO-2020124515-A1 QUINOLINE DERIVATIVE, PREPARATION METHOD AND USE THEREOF 东莞市东阳光农药研发有限公司 2020-06-25 WO disclosed