SCHEMBL2223699

SCHEMBL2223699

Cc1ccc(F)cc1Oc1ncc2nc(-c3cc(C)c([O])c(C)c3)oc2n1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.45
CEPT1 Q9Y6K0 2/20 0.36
TP53 P04637 1/20 0.36
THRB P10828 1/20 0.36
APP P05067 9/20 0.35
PDGFRB P09619 1/20 0.34
PDGFRA P16234 1/20 0.34
MAOB P27338 2/20 0.33
CETP P11597 2/20 0.33
RXFP1 Q9HBX9 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
HIF1A Q16665 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2223599 0.93 S1PR1 (0.47) S1PR1CEPT1TP53THRBAPP
SCHEMBL2223206 0.91 S1PR1 (0.47) S1PR1CEPT1APPMAOBUSP2
SCHEMBL2222292 0.91 S1PR1 (0.44) S1PR1
SCHEMBL2224142 0.89 S1PR1 (0.51) S1PR1TP53APPCETPRXFP1
SCHEMBL2224913 0.89 S1PR1 (0.47) S1PR1CEPT1APPCETPALDH1A1
SCHEMBL2222186 0.88 S1PR1 (0.48) S1PR1CEPT1TP53THRBAPP
SCHEMBL2224919 0.88 S1PR1 (0.49) S1PR1CEPT1TP53THRBCETP
SCHEMBL2224286 0.87 S1PR1 (0.54) S1PR1CEPT1TP53THRBAPP
SCHEMBL2225559 0.86 S1PR1 (0.49) S1PR1CEPT1TP53THRBAPP
SCHEMBL14797212 0.85 S1PR1 (0.66) S1PR1CEPT1TP53THRBCETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011086079-A1 CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING SANOFI-AVENTIS (FR) 2011-07-21 WO disclosed