SCHEMBL22258784

SCHEMBL22258784

CN(CC1CCCCC1)C(=O)c1c[nH]nc1-c1ccncc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.36
MAPK1 P28482 2/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
PRSS12 P56730 1/20 0.35
CDC7 O00311 1/20 0.34
MELK Q14680 2/20 0.34
BUB1 O43683 1/20 0.34
CYP19A1 P11511 2/20 0.34
KDM4C Q9H3R0 1/20 0.33
DYRK1A Q13627 1/20 0.33
MAPK11 Q15759 1/20 0.33
MAPK14 Q16539 1/20 0.33
PAX8 Q06710 1/20 0.33
SLC2A1 P11166 1/20 0.33
NAMPT P43490 1/20 0.33
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22258961 0.77 CNR1 (0.47) POLBKDM4CNAMPT
SCHEMBL22258955 0.73 CYP19A1 (0.33) MAPK1ALDH1A1CDC7CYP19A1MAPK11
SCHEMBL31098460 0.70 SMN1; SMN2 (0.47) TSHRALDH1A1MEN1KMT2A
SCHEMBL22258783 0.70 CSNK1A1 (0.42) MAPK1ALDH1A1POLBCDC7MAPK14
SCHEMBL22258956 0.64 ROCK2 (0.44) MAPK1MELKDYRK1A
SCHEMBL22258664 0.64 CHEK1 (0.57) MAPK1
SCHEMBL22258786 0.64 CSNK2A2 (0.48) DYRK1A
SCHEMBL5946809 0.63 PDK1 (0.44) PDK1PDK2PDK3PDK4
SCHEMBL31098537 0.63 ALDH1A1 (0.46) ALDH1A1KMT2A
SCHEMBL22554282 0.63 PAX8 (0.42) TSHRALDH1A1MELKMAPK14PAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020150545-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF THE WNT/B-CATENIN SIGNALING PATHWAY SAMUMED, LLC (US) 2020-07-23 WO disclosed