SCHEMBL22322334

SCHEMBL22322334

COc1cc(C=O)cnc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.50
MAPT P10636 6/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
FDPS P14324 1/20 0.50
TSHR P16473 1/20 0.48
GAA P10253 1/20 0.46
HPGD P15428 3/20 0.44
TRIM24 O15164 1/20 0.44
ALDH5A1 P51649 1/20 0.44
ABAT P80404 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
TRIM33 Q9UPN9 1/20 0.44
CYP1A2 P05177 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2D6 P10635 1/20 0.43
MAPK1 P28482 1/20 0.43
LMNA P02545 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29954141 1.00 ALDH1A1 (0.50) ALDH1A1MAPTMEN1KMT2AFDPS
SCHEMBL23905081 0.80 ALDH1A1 (0.45) ALDH1A1MAPTMEN1KMT2AFDPS
SCHEMBL29936033 0.79 FDPS (0.51) ALDH1A1MAPTMEN1KMT2AFDPS
SCHEMBL25355441 0.79 FDPS (0.51) ALDH1A1MAPTMEN1KMT2AFDPS
SCHEMBL29950972 0.79 FDPS (0.51) ALDH1A1MAPTMEN1KMT2AFDPS
SCHEMBL2698927 0.79 FDPS (0.51) ALDH1A1MAPTMEN1KMT2AFDPS
SCHEMBL13723899 0.78 FDPS (0.50) ALDH1A1MAPTMEN1KMT2AFDPS
SCHEMBL16564249 0.78 ALDH1A1 (0.53) ALDH1A1MAPTMEN1KMT2AFDPS
SCHEMBL29954529 0.78 FDPS (0.50) ALDH1A1MAPTMEN1KMT2AFDPS
SCHEMBL10131337 0.78 FDPS (0.50) ALDH1A1MAPTMEN1KMT2AFDPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12612407-B2 Imidazo[2,1-f][1,2,4]triazin-4-amine derivatives as TLR7 agonist BEONE MEDICINES I GMBH (CH) 2026-04-28 US disclosed
CN-113423708-B Imidazo [2,1-F ] [1,2,4] triazin-4-amine derivatives as TLR7 agonists 百济神州有限公司 2025-04-22 CN disclosed
EP-3921319-B1 IMIDAZO [2, 1-F] [1, 2, 4] TRIAZIN-4-AMINE DERIVATIVES AS TLR7 AGONIST BEIGENE LTD (KY) 2024-03-06 EP disclosed
US-20230167117-A1 IMIDAZO[2,1-F][1,2,4]TRIAZIN-4-AMINE DERIVATIVES AS TLR7 AGONIST BEONE MEDICINES I GMBH (CH) 2023-06-01 US disclosed
US-20220281873-A1 COMPOUND AS PORCUPINE INHIBITOR AND USE THEREOF MEDSHINE DISCOVERY INC. (CN) 2022-09-08 US disclosed
EP-3921319-A1 IMIDAZO [2, 1-F] [1, 2, 4] TRIAZIN-4-AMINE DERIVATIVES AS TLR7 AGONIST BeiGene, Ltd. (KY) 2021-12-15 EP disclosed
CN-113423708-A Imidazo [2,1-F ] [1,2,4] triazin-4-amine derivatives as TLR7 agonists 百济神州有限公司 2021-09-21 CN disclosed
WO-2021004467-A1 COMPOUND AS PORCUPINE INHIBITOR AND USE THEREOF 南京明德新药研发有限公司 2021-01-14 WO disclosed
WO-2020160710-A1 IMIDAZO [2, 1-F] [1, 2, 4] TRIAZIN-4-AMINE DERIVATIVES AS TLR7 AGONIST BEIGENE, LTD. (KY) 2020-08-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220281873-A1 COMPOUND AS PORCUPINE INHIBITOR AND USE THEREOF PORCN, SLC6A1, SLC6A11 ALDH1A1 2067/4885MAPT 683/4885MEN1 1480/4885
US-20230167117-A1 IMIDAZO[2,1-F][1,2,4]TRIAZIN-4-AMINE DERIVATIVES AS TLR7 AGONIST TLR7, TLR1, TLR9 ALDH1A1 1537/4885MAPT 3947/4885MEN1 2941/4885
US-12612407-B2 Imidazo[2,1-f][1,2,4]triazin-4-amine derivatives as TLR7 agonist TLR7, TLR8, TLR1 ALDH1A1 1253/4885MAPT 4628/4885MEN1 4551/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.