SCHEMBL22353633

SCHEMBL22353633

COC(=O)C12CCCC(C1)C(C#N)CC2

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
TSHR P16473 1/20 0.30
CYP2C19 P33261 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27444382 0.76 HSD11B1 (0.30)
SCHEMBL19189061 0.76 SLC6A12 (0.34) TSHRNPSR1MAPT
SCHEMBL23329861 0.75 CYP4F2 (0.33) NPSR1MAPT
SCHEMBL25074421 0.75 EPHX1 (0.33) NPSR1MAPT
SCHEMBL9951753 0.72 NPSR1 (0.38) TSHRNPSR1MAPT
SCHEMBL22824391 0.70 KCNA3 (0.31)
SCHEMBL14299766 0.70 PKM (0.39)
SCHEMBL3704482 0.68 ALDH1A1 (0.42) TSHRNPSR1MAPT
SCHEMBL22354094 0.66 HSD11B1 (0.33)
SCHEMBL25747292 0.66 GAA (0.33) CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020168143-A1 SUBSTITUTED BICYCLIC COMPOUNDS AS FARNESOID X RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2020-08-20 WO disclosed