SCHEMBL22354094

SCHEMBL22354094

COC(=O)C12CCCC(C1)C(c1ncc(Br)cn1)CC2

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.33
OPRK1 P41145 8/20 0.32
HCRTR2 O43614 2/20 0.31
DGAT1 O75907 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22347663 0.68 HSD11B1 (0.39) HSD11B1OPRK1DGAT1NPC1RAB9A
SCHEMBL19189061 0.68 SLC6A12 (0.34)
SCHEMBL25074421 0.67 EPHX1 (0.33)
SCHEMBL23329861 0.67 CYP4F2 (0.33)
SCHEMBL22353633 0.66 DPP4 (0.30)
SCHEMBL9951753 0.65 NPSR1 (0.38)
SCHEMBL14968320 0.64 HSD11B1 (0.35) HSD11B1OPRK1DGAT1NPC1RAB9A
SCHEMBL22824391 0.63 KCNA3 (0.31)
SCHEMBL13769236 0.62 LMNA (0.34)
SCHEMBL1282303 0.61 OPRK1 (0.38) OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020168143-A1 SUBSTITUTED BICYCLIC COMPOUNDS AS FARNESOID X RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2020-08-20 WO disclosed