SCHEMBL2250684

SCHEMBL2250684

COc1cccc(-c2ccccc2COc2ccc(-c3ccc(C(=O)N[C@@H](CCC(N)=O)C(=O)O)cc3)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.46
KMT2A Q03164 2/20 0.46
GAA P10253 1/20 0.46
PTGER4 P35408 3/20 0.46
PTGER3 P43115 2/20 0.46
PTGER1 P34995 1/20 0.46
PTGER2 P43116 1/20 0.46
FFAR1 O14842 2/20 0.46
FFAR4 Q5NUL3 2/20 0.46
CA2 P00918 2/20 0.44
ALDH1A1 P00352 2/20 0.44
CTDSP1 Q9GZU7 1/20 0.44
CA1 P00915 1/20 0.44
PTPN1 P18031 1/20 0.44
CD274 Q9NZQ7 4/20 0.44
TRPV1 Q8NER1 1/20 0.43
C3AR1 Q16581 1/20 0.43
CYP3A4 P08684 1/20 0.42
MRGPRX4 Q96LA9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2251027 0.90 CA2 (0.51) FFAR1FFAR4CA2CA1PTPN1
SCHEMBL2250678 0.90 MMP12 (0.54) POLBKMT2AGAAPTGER4PTGER3
SCHEMBL2250715 0.87 MRGPRX4 (0.51) POLBKMT2AGAAFFAR1CA2
SCHEMBL2245262 0.87 MRGPRX4 (0.53) POLBKMT2AGAACA2ALDH1A1
SCHEMBL3589157 0.83 KLKB1 (0.50) PTGER4PTGER3PTGER1PTGER2FFAR1
SCHEMBL2243990 0.82 DHFR (0.50) POLBKMT2AGAACA2ALDH1A1
SCHEMBL2247651 0.81 MRGPRX4 (0.56) FFAR1FFAR4CA2CA1MRGPRX4
SCHEMBL3589161 0.80 HSD17B2 (0.45) KMT2APTGER4PTGER3PTGER1PTGER2
SCHEMBL2251677 0.80 GPR132 (0.55) FFAR1CA2ALDH1A1CA1PTPN1
SCHEMBL2251026 0.79 MMP12 (0.57) PTGER4PTGER3PTGER1PTGER2FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed