SCHEMBL22453357

SCHEMBL22453357

CN(c1ccc(C(F)(F)F)cc1)c1ccc(N)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.41
ALDH1A1 P00352 3/20 0.38
POLQ O75417 1/20 0.35
TAAR1 Q96RJ0 1/20 0.34
SCN9A Q15858 1/20 0.34
PKM P14618 1/20 0.33
BACE1 P56817 1/20 0.33
CFTR P13569 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
GAA P10253 1/20 0.33
LTC4S Q16873 1/20 0.33
PDK2 Q15119 1/20 0.33
RAB9A P51151 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PTGS1 P23219 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22453355 0.83 S100B (0.50) KIF11ALDH1A1SCN9APKMBACE1
SCHEMBL13367596 0.80 KIF11 (0.50) KIF11ALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL22453522 0.80 DHFR (0.44) KIF11ALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL22453358 0.79 MAPT (0.41) ALDH1A1SCN9AKDM4EHSD17B10RAB9A
SCHEMBL22453192 0.78 KIF11 (0.59) KIF11ALDH1A1TAAR1L3MBTL1PTGS1
SCHEMBL22452606 0.77 ALDH1A1 (0.38) ALDH1A1
SCHEMBL379155 0.76 ALDH1A1 (0.52) KIF11ALDH1A1PKMBACE1CFTR
SCHEMBL17504172 0.75 MTOR (0.42) KIF11POLQSCN9ALTC4SPDK2
Hydrochloric Acid SCHEMBL30779699 0.74 IDO1 (0.52) KIF11ALDH1A1PKMBACE1CFTR
Bromide SCHEMBL29950269 0.74 ALDH1A1 (0.50) KIF11ALDH1A1PKMBACE1CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed