SCHEMBL22453358

SCHEMBL22453358

CN(c1ccc(OCC(F)(F)F)cc1)c1ccc(N)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.41
ALDH1A1 P00352 4/20 0.41
KDM4C Q9H3R0 2/20 0.40
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
KDM4E B2RXH2 2/20 0.38
USP2 O75604 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
THRB P10828 1/20 0.38
G6PD P11413 1/20 0.38
ALOX15 P16050 1/20 0.38
CASP1 P29466 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP2C9 P11712 2/20 0.35
CYP17A1 P05093 1/20 0.35
CYP2C19 P33261 1/20 0.35
CYP1A2 P05177 1/20 0.35
LMNA P02545 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22452931 0.86 S100B (0.46) MAPTALDH1A1KDM4CMEN1KMT2A
SCHEMBL22452587 0.82 ALDH1A1 (0.49) MAPTALDH1A1KDM4CMEN1KMT2A
SCHEMBL22453522 0.81 DHFR (0.44) ALDH1A1KDM4CGPR3DHFR
SCHEMBL22453357 0.79 KIF11 (0.41) ALDH1A1L3MBTL1KDM4EHSD17B10SCN9A
SCHEMBL22681911 0.74 KDM4C (0.40) MAPTALDH1A1KDM4CMEN1KMT2A
SCHEMBL22452606 0.70 ALDH1A1 (0.38) ALDH1A1
SCHEMBL498377 0.69 ALDH1A1 (0.56) MAPTALDH1A1MEN1KMT2AL3MBTL1
Hydrochloric Acid SCHEMBL9530875 0.69 ALDH1A1 (0.55) MAPTALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL12021921 0.68 BRD4 (0.40) MAPTALDH1A1MEN1KMT2ACYP2C9
SCHEMBL9682 0.68 MAPT (0.63) MAPTALDH1A1MEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed