SCHEMBL2247526

SCHEMBL2247526

NC(=O)[C@H](CCC(=O)O)NC(=O)c1ccc(-c2ccco2)cc1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 3/20 0.58
HPGDS O60760 4/20 0.55
CA1 P00915 2/20 0.50
CA12 O43570 1/20 0.50
CA9 Q16790 1/20 0.50
PTPN1 P18031 1/20 0.48
ADAMTS5 Q9UNA0 2/20 0.47
ADAMTS4 O75173 1/20 0.47
CA2 P00918 2/20 0.47
MMP2 P08253 2/20 0.43
MMP8 P22894 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
LMNA P02545 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HDAC2 Q92769 1/20 0.43
TAAR1 Q96RJ0 1/20 0.42
PPARD Q03181 1/20 0.42
FOLH1 Q04609 1/20 0.41
PDE4A P27815 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2247532 0.86 CA2 (0.58) MMP12CA1CA2MMP2HDAC2
SCHEMBL2246054 0.85 MMP12 (0.76) MMP12HPGDSCA1CA12CA9
SCHEMBL2245321 0.85 MMP12 (0.76) MMP12HPGDSCA1CA12CA9
SCHEMBL2245742 0.82 PTPN2 (0.56) MMP12HPGDSPTPN1
SCHEMBL3579193 0.82 ADAMTS5 (0.50) MMP12ADAMTS5ADAMTS4MMP2MMP8
SCHEMBL28108803 0.80 HPGDS (0.69) MMP12HPGDSCA1CA12CA9
SCHEMBL10518630 0.80 HPGDS (0.69) MMP12HPGDSCA1CA12CA9
SCHEMBL2247335 0.80 C3AR1 (0.46) MMP12HPGDSPTPN1MMP2MMP8
SCHEMBL2245606 0.80 MMP12 (0.65) MMP12HPGDSCA1CA12CA9
SCHEMBL2248624 0.78 MMP12 (0.64) MMP12HPGDSCA1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed