SCHEMBL2248592

SCHEMBL2248592

NC(=O)CC[C@H](NC(=O)c1ccc(-c2ccc(OCc3ccc4ccccc4c3)cc2)cc1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.54
PTPN1 P18031 3/20 0.53
NPC1 O15118 1/20 0.51
MAPT P10636 1/20 0.51
CA2 P00918 3/20 0.51
FPGS Q05932 2/20 0.50
MRGPRX4 Q96LA9 1/20 0.50
PTPN2 P17706 1/20 0.49
CDC25B P30305 1/20 0.49
ADAMTS4 O75173 1/20 0.49
MMP13 P45452 1/20 0.49
CTSL P07711 1/20 0.49
CTSB P07858 1/20 0.49
CTSS P25774 1/20 0.49
CTSK P43235 1/20 0.49
CA1 P00915 1/20 0.49
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
GPR132 Q9UNW8 1/20 0.48
PIN1 Q13526 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2247651 0.90 MRGPRX4 (0.56) DHFRCA2FPGSMRGPRX4CA1
SCHEMBL2251677 0.90 GPR132 (0.55) DHFRPTPN1MAPTCA2MRGPRX4
SCHEMBL2248588 0.88 MMP12 (0.57) DHFRPTPN1NPC1MAPTCA2
SCHEMBL2249558 0.86 CA2 (0.58) PTPN1CA2CTSLCTSBCTSS
SCHEMBL2246956 0.85 GRM5 (0.57) DHFRCA2MRGPRX4ADAMTS4MMP13
SCHEMBL2247421 0.85 PARP15 (0.56) DHFRNPC1CA2FPGSMRGPRX4
SCHEMBL2245262 0.85 MRGPRX4 (0.53) DHFRPTPN1NPC1CA2FPGS
SCHEMBL2243990 0.83 DHFR (0.50) DHFRPTPN1MAPTCA2FPGS
SCHEMBL2250715 0.83 MRGPRX4 (0.51) DHFRPTPN1NPC1CA2MRGPRX4
SCHEMBL2251027 0.82 CA2 (0.51) DHFRPTPN1CA2PTPN2CDC25B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed