SCHEMBL22492843

SCHEMBL22492843

CC(C)[Si](C#Cc1cccc(Nc2ccsc2C(=O)c2ccccc2)c1)(C(C)C)C(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 3/20 0.38
GRM5 P41594 1/20 0.37
MAPT P10636 3/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
ALK Q9UM73 6/20 0.37
CCNA2 P20248 2/20 0.36
CDK2 P24941 2/20 0.36
PKM P14618 1/20 0.35
PTPN11 Q06124 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CSNK2A2 P19784 1/20 0.35
CSNK2B P67870 1/20 0.35
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
MAPK14 Q16539 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22492821 0.81 CSNK2A1 (0.49) CSNK2A1MAPTALDH1A1L3MBTL1
SCHEMBL22492839 0.81 CSNK2A1 (0.49) CSNK2A1NPC1RAB9ACCNA2CDK2
SCHEMBL2798077 0.77 ALDH1A1 (0.50) MAPTRAB9AALDH1A1PTPN11L3MBTL1
SCHEMBL22492805 0.75 CDK2 (0.57) CSNK2A1MAPTNPC1RAB9AALDH1A1
SCHEMBL22492833 0.75 SIRT2 (0.48) MAPTNPC1RAB9ACCNA2CDK2
SCHEMBL22492801 0.74 MAPT (0.59) CSNK2A1MAPTNPC1RAB9AALDH1A1
SCHEMBL22492828 0.71 CCNA2 (0.52) CSNK2A1MAPTNPC1RAB9AALDH1A1
SCHEMBL22492764 0.70 RAB9A (0.52) MAPTNPC1RAB9AALDH1A1POLB
SCHEMBL16346233 0.69 ACACB (0.50) GRM5NPC1RAB9AALDH1A1ALK
SCHEMBL26988072 0.68 LMNA (0.40) MAPTRAB9AALDH1A1ALKL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210188763-A1 COMPOUNDS AND METHODS FOR HEMATOPOIETIC REGENERATION UNIV CALIFORNIA (US) 2021-06-24 US disclosed
EP-3717450-A1 COMPOUNDS AND METHODS FOR HEMATOPOIETIC REGENERATION The Regents of the University of California (US) 2020-10-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210188763-A1 COMPOUNDS AND METHODS FOR HEMATOPOIETIC REGENERATION HGF, CXCL12, CCL11 CSNK2A1 3987/4885GRM5 3579/4885MAPT 4809/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.