SCHEMBL31407

SCHEMBL31407

O=C(c1cccc(O)c1)c1nc2ccccc2s1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 8/20 0.79
HSD17B2 P37059 7/20 0.79
DYRK1A Q13627 2/20 0.58
FAAH O00519 1/20 0.54
CYP1A2 P05177 2/20 0.53
CYP3A4 P08684 2/20 0.53
CYP2D6 P10635 2/20 0.53
CYP2C9 P11712 2/20 0.53
CYP2B6 P20813 2/20 0.53
CYP2C19 P33261 2/20 0.53
LMNA P02545 1/20 0.52
TP53 P04637 1/20 0.52
POLB P06746 1/20 0.52
NFKB1 P19838 1/20 0.52
RAB9A P51151 1/20 0.52
NFKB2 Q00653 1/20 0.52
RELA Q04206 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
HSD17B10 Q99714 1/20 0.52
BCL2 P10415 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29786 0.88 HSD17B1 (1.00) HSD17B1HSD17B2DYRK1ACYP1A2CYP3A4
SCHEMBL24751 0.84 HSD17B1 (0.62) HSD17B1HSD17B2LMNATP53NFKB1
SCHEMBL900711 0.84 SCD (0.62) HSD17B1HSD17B2FAAHCYP1A2CYP3A4
SCHEMBL27623260 0.84 HSD17B1 (0.67) HSD17B1HSD17B2FAAHCYP1A2CYP3A4
SCHEMBL1304947 0.83 HSD17B1 (0.66) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
Bromide SCHEMBL28862925 0.83 HSD17B1 (0.61) HSD17B1HSD17B2LMNATP53NFKB1
SCHEMBL31078 0.81 RAB9A (0.65) HSD17B1HSD17B2FAAHLMNATP53
SCHEMBL8400538 0.81 HSD17B1 (0.81) HSD17B1HSD17B2DYRK1ACYP1A2CYP3A4
SCHEMBL6319718 0.81 ALDH1A1 (0.66) HSD17B1HSD17B2DYRK1ALMNATP53
SCHEMBL8405370 0.80 HSD17B1 (0.74) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP claimed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO claimed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed
WO-2008129129-A1 HETEROCYCLIC PHENYL CARBAMATES AS NOVEL FAAH-INHIBITORS KUOPION YLIOPISTO (FI) 2008-10-30 WO disclosed