SCHEMBL22561920

SCHEMBL22561920

Cc1cnc(S(C)(=O)=O)c(C#N)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35
MAPT P10636 1/20 0.35
LRRK2 Q5S007 9/20 0.35
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
SCN9A Q15858 1/20 0.32
SLC22A12 Q96S37 1/20 0.32
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethyl Sulfone SCHEMBL17258778 0.81 NOS3 (0.46) KMT2AKDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL17591619 0.81 KMT2A (0.38) KMT2AKDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL27416291 0.77 XDH (0.44) ALDH1A1HPGD
SCHEMBL14159470 0.76 ALDH1A1 (0.56) KMT2AKDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL31108446 0.76 CYP11B2 (0.40) KMT2AKDM4ELMNASMN1; SMN2MAPT
SCHEMBL15047723 0.75 NOS3 (0.45) KMT2AKDM4EALDH1A1LMNACYP1A2
SCHEMBL21048809 0.75 GAA (0.33) KDM4EALDH1A1HTTLRRK2CYP11B1
SCHEMBL1626886 0.73 PTK2 (0.37) KDM4EALDH1A1HTTLRRK2
SCHEMBL27465877 0.73 POLB (0.38) LRRK2SCN9A
SCHEMBL625135 0.73 NOS3 (0.54) KMT2AKDM4EALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3191467-B1 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS NOVARTIS AG (CH) 2020-10-21 EP disclosed