SCHEMBL22604347

SCHEMBL22604347

C=C1C(c2ccc3c(c2)C=CC(C)(C)O3)=CCc2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 9/20 0.36
EPAS1 Q99814 9/20 0.36
PPARG P37231 2/20 0.33
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
CA12 O43570 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CA1 P00915 1/20 0.32
TP53 P04637 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
CA7 P43166 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CA9 Q16790 1/20 0.32
CA13 Q8N1Q1 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8902134 0.67 HIF1A (0.39) HIF1AEPAS1PPARGKDM4ENPC1
SCHEMBL20124031 0.66 MAOA (0.42) KDM4ENPC1ALDH1A1MAPTHPGD
SCHEMBL9475843 0.64 ALDH1A1 (0.45) HIF1AEPAS1KDM4ENPC1CA12
SCHEMBL9092301 0.64 HIF1A (0.48) HIF1AEPAS1ALDH1A1HPGD
SCHEMBL1748567 0.63 HTR2C (0.49) HIF1AEPAS1KDM4ENPC1CA12
SCHEMBL29644871 0.63 HTR2C (0.49) HIF1AEPAS1KDM4ENPC1CA12
SCHEMBL3049240 0.62 ALDH1A1 (0.46) HIF1AEPAS1KDM4ENPC1CA12
SCHEMBL7738844 0.62 HIF1A (0.58) HIF1AEPAS1KDM4ENPC1CA12
SCHEMBL9092974 0.62 HIF1A (0.46) HIF1AEPAS1KDM4ENPC1CA12
SCHEMBL9092213 0.62 HIF1A (0.44) HIF1AEPAS1KDM4ENPC1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020215481-A1 APPLICATIONS OF PSORALEN IN PREPARING NRF2 INHIBITOR, MEDICAMENT FOR NRF2 INHIBITION-RELATED DISEASES, AND ANTICANCER MEDICAMENT 广东省中医院 2020-10-29 WO disclosed