SCHEMBL22632891

SCHEMBL22632891

Cc1ccc(S(=O)(=O)n2cc(C(C)C)c3nc(Cc4c(C)cc(N)cc4C)cnc32)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.34
HTR6 P50406 3/20 0.32
MAPT P10636 2/20 0.32
ALDH1A1 P00352 2/20 0.32
KLKB1 P03952 1/20 0.32
KDM4E B2RXH2 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TSHR P16473 1/20 0.31
ALK Q9UM73 1/20 0.31
PTPN11 Q06124 1/20 0.31
POLB P06746 1/20 0.31
ALDH3A1 P30838 1/20 0.31
HTT P42858 1/20 0.31
NOD1 Q9Y239 1/20 0.31
MBOAT4 Q96T53 1/20 0.31
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22632665 0.91 ALK (0.35) L3MBTL1HTR6MAPTALDH1A1KDM4E
SCHEMBL22632745 0.88 L3MBTL1 (0.32) L3MBTL1ALDH1A1TSHRALKPTPN11
SCHEMBL22638209 0.87 PDE4A (0.35) L3MBTL1ALDH1A1KLKB1GAATSHR
SCHEMBL29414678 0.85 PTGS2 (0.32) L3MBTL1PTPN11HTT
SCHEMBL22632642 0.85 PTGS2 (0.32) L3MBTL1PTPN11HTT
SCHEMBL22632544 0.85 ALK (0.36) L3MBTL1HTR6MAPTALDH1A1KLKB1
SCHEMBL22632786 0.84 CD4 (0.42) L3MBTL1HTR6ALDH1A1ALK
SCHEMBL22633321 0.84 L3MBTL1 (0.30) L3MBTL1
SCHEMBL31258414 0.84 CD4 (0.42) L3MBTL1HTR6ALDH1A1ALK
SCHEMBL29414769 0.84 L3MBTL1 (0.30) L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122036699-A THR-beta modulators and methods of use thereof 阿利戈斯治疗公司 2026-05-15 CN disclosed
US-20250304561-A1 MODULATORS OF THR-BETA AND METHODS OF USE THEREOF ALIGOS THERAPEUTICS, INC. (US) 2025-10-02 US disclosed
EP-4523692-A2 MODULATORS OF THR-SS AND METHODS OF USE THEREOF Aligos Therapeutics, Inc. (US) 2025-03-19 EP disclosed
EP-3965884-B1 MODULATORS OF THR-BETA WITH A DIOXO-1,2,4-TRIAZYL HEAD GROUP ALIGOS THERAPEUTICS INC (US) 2025-01-15 EP disclosed
US-12180192-B2 Modulators of THR-β and methods of use thereof ALIGOS THERAPEUTICS, INC. (US) 2024-12-31 US disclosed
US-20210355112-A1 MODULATORS OF THR-BETA AND METHODS OF USE THEREOF ALIGOS THERAPEUTICS, INC. (US) 2021-11-18 US disclosed
US-11091467-B2 Modulators of THR-β and methods of use thereof ALIGOS THERAPEUTICS, INC. (US) 2021-08-17 US disclosed
US-20200354345-A1 MODULATORS OF THR-BETA AND METHODS OF USE THEREOF ALIGOS THERAPEUTICS, INC. (US) 2020-11-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210355112-A1 MODULATORS OF THR-BETA AND METHODS OF USE THEREOF THRB, THRA, TRHR L3MBTL1 527/4885HTR6 710/4885MAPT 1399/4885
US-20250304561-A1 MODULATORS OF THR-BETA AND METHODS OF USE THEREOF THRB, THRA, TRHR L3MBTL1 1414/4885HTR6 945/4885MAPT 1383/4885
US-20200354345-A1 MODULATORS OF THR-BETA AND METHODS OF USE THEREOF THRB, THRA, TRHR L3MBTL1 527/4885HTR6 710/4885MAPT 1399/4885
US-12180192-B2 Modulators of THR-β and methods of use thereof THRB, THRA, TRHR L3MBTL1 798/4885HTR6 765/4885MAPT 1243/4885
US-11091467-B2 Modulators of THR-β and methods of use thereof THRB, THRA, TRHR L3MBTL1 798/4885HTR6 765/4885MAPT 1243/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.