SCHEMBL22643113

SCHEMBL22643113

CCc1ccc(-n2cc(CC(O)C(C)C)nn2)cc1F

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.54
CTSC P53634 3/20 0.54
RXRA P19793 12/20 0.47
GRIN1 Q05586 11/20 0.47
GRIN2B Q13224 11/20 0.47
ALDH1A1 P00352 1/20 0.46
KCNH2 Q12809 1/20 0.44
DPP4 P27487 1/20 0.43
DDX3X O00571 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22642979 0.80 NOTUM (0.60) CTSKCTSCRXRAGRIN1GRIN2B
SCHEMBL22643118 0.79 P2RX7 (0.60) CTSKCTSCRXRAGRIN1GRIN2B
SCHEMBL22643391 0.75 KCNH2 (0.58) CTSKCTSCRXRAGRIN1GRIN2B
SCHEMBL22643248 0.74 CTSK (0.55) CTSKCTSCRXRAGRIN1GRIN2B
SCHEMBL22643453 0.74 KCNH2 (0.57) CTSKCTSCRXRAGRIN1GRIN2B
SCHEMBL22643285 0.74 CTSK (0.49) CTSKCTSCRXRAGRIN1GRIN2B
SCHEMBL22643110 0.73 CA9 (0.51) CTSKCTSCRXRAGRIN1GRIN2B
SCHEMBL16064307 0.72 CTSC (1.00) CTSKCTSC
SCHEMBL19220682 0.70 RXRA (0.69) RXRAGRIN1GRIN2BKCNH2
SCHEMBL30031099 0.70 NOTUM (0.50) RXRAGRIN1GRIN2BKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970283-B1 SUBSTITUTED 2-AZA-BICYCLO[2.2.1]HEPTANE-3-CARBOXYLIC ACID (BENZYL-CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C BOEHRINGER INGELHEIM INT (DE) 2020-11-11 EP disclosed