SCHEMBL22643285

SCHEMBL22643285

CCc1ccc(-n2cc(C(C)=O)nn2)cc1F

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.49
CTSC P53634 1/20 0.49
KMT2A Q03164 1/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ESRRA P11474 2/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
RXRA P19793 4/20 0.41
GRIN1 Q05586 4/20 0.41
GRIN2B Q13224 4/20 0.41
NOTUM Q6P988 2/20 0.41
MIF P14174 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14701729 0.78 CA1 (0.56) KMT2ANPC1RAB9ASMN1; SMN2ESRRA
SCHEMBL20263181 0.77 KMT2A (0.50) KMT2ANPC1RAB9ASMN1; SMN2ESRRA
SCHEMBL22643110 0.75 CA9 (0.51) CTSKCTSCCA12CA1CA2
SCHEMBL22642979 0.75 NOTUM (0.60) CTSKCTSCRXRAGRIN1GRIN2B
SCHEMBL22643118 0.74 P2RX7 (0.60) CTSKCTSCRXRAGRIN1GRIN2B
SCHEMBL22643113 0.74 CTSK (0.54) CTSKCTSCALDH1A1RXRAGRIN1
SCHEMBL22643248 0.72 CTSK (0.55) CTSKCTSCKMT2ANPC1ALDH1A1
SCHEMBL23889183 0.71 ESRRA (0.59) NPC1ESRRACA1CA2CA9
SCHEMBL30412575 0.71 SIGMAR1 (0.39) KMT2ARXRAGRIN1GRIN2B
SCHEMBL24215708 0.71 SIGMAR1 (0.39) KMT2ARXRAGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970283-B1 SUBSTITUTED 2-AZA-BICYCLO[2.2.1]HEPTANE-3-CARBOXYLIC ACID (BENZYL-CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C BOEHRINGER INGELHEIM INT (DE) 2020-11-11 EP disclosed