SCHEMBL22643118

SCHEMBL22643118

CCOCc1cn(-c2ccc(CC)c(F)c2)nn1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.60
RXRA P19793 15/20 0.56
GRIN1 Q05586 15/20 0.56
GRIN2B Q13224 15/20 0.56
DDX3X O00571 3/20 0.53
CTSK P43235 1/20 0.51
CTSC P53634 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22642979 0.88 NOTUM (0.60) RXRAGRIN1GRIN2BCTSKCTSC
SCHEMBL22643248 0.79 CTSK (0.55) P2RX7RXRAGRIN1GRIN2BCTSK
SCHEMBL22643113 0.79 CTSK (0.54) RXRAGRIN1GRIN2BDDX3XCTSK
SCHEMBL22643110 0.75 CA9 (0.51) RXRAGRIN1GRIN2BCTSKCTSC
SCHEMBL17978485 0.75 P2RX7 (0.74) P2RX7RXRAGRIN1GRIN2BDDX3X
SCHEMBL15316360 0.75 P2RX7 (0.73) P2RX7RXRAGRIN1GRIN2BDDX3X
SCHEMBL21974270 0.75 RXRA (0.68) P2RX7RXRAGRIN1GRIN2BDDX3X
SCHEMBL29828653 0.74 P2RX7 (0.67) P2RX7DDX3X
SCHEMBL22643285 0.74 CTSK (0.49) RXRAGRIN1GRIN2BCTSKCTSC
SCHEMBL17978607 0.73 P2RX7 (0.65) P2RX7DDX3X

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970283-B1 SUBSTITUTED 2-AZA-BICYCLO[2.2.1]HEPTANE-3-CARBOXYLIC ACID (BENZYL-CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C BOEHRINGER INGELHEIM INT (DE) 2020-11-11 EP disclosed