SCHEMBL22643248

SCHEMBL22643248

CCc1ccc(-n2cc(COC(=O)N3CCCC3)nn2)cc1F

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.55
CTSC P53634 1/20 0.55
ALDH1A1 P00352 1/20 0.49
RXRA P19793 11/20 0.48
GRIN1 Q05586 11/20 0.48
GRIN2B Q13224 11/20 0.48
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
HPGD P15428 1/20 0.43
NPC1 O15118 2/20 0.43
KMT2A Q03164 1/20 0.43
P2RX7 Q99572 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22642979 0.81 NOTUM (0.60) CTSKCTSCRXRAGRIN1GRIN2B
SCHEMBL22643118 0.79 P2RX7 (0.60) CTSKCTSCRXRAGRIN1GRIN2B
SCHEMBL22643113 0.74 CTSK (0.54) CTSKCTSCALDH1A1RXRAGRIN1
SCHEMBL16064249 0.73 CTSC (1.00) CTSKCTSC
SCHEMBL22643285 0.72 CTSK (0.49) CTSKCTSCALDH1A1RXRAGRIN1
SCHEMBL22643110 0.69 CA9 (0.51) CTSKCTSCRXRAGRIN1GRIN2B
SCHEMBL30031099 0.66 NOTUM (0.50) RXRAGRIN1GRIN2BP2RX7
SCHEMBL21737191 0.66 MAPT (0.45) ALDH1A1HPGDNPC1KMT2A
SCHEMBL543019 0.65 ENPP2 (0.52) ALDH1A1CYP2D6HPGDKMT2A
SCHEMBL19219658 0.65 RXRA (1.00) RXRAGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970283-B1 SUBSTITUTED 2-AZA-BICYCLO[2.2.1]HEPTANE-3-CARBOXYLIC ACID (BENZYL-CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C BOEHRINGER INGELHEIM INT (DE) 2020-11-11 EP disclosed