SCHEMBL22650515

SCHEMBL22650515

COc1nc(-c2ccnc(Nc3ccc(N4CCCC(N(C)C)C4=O)cc3)n2)cc2c1ncn2C(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 7/20 0.35
JAK2 O60674 4/20 0.35
BRD4 O60885 5/20 0.34
CDK9 P50750 4/20 0.34
CDK1 P06493 1/20 0.34
CDK4 P11802 1/20 0.34
CCNB1 P14635 1/20 0.34
CCND1 P24385 1/20 0.34
JAK3 P52333 1/20 0.33
IKBKB O14920 1/20 0.33
CHUK O15111 1/20 0.33
IKBKG Q9Y6K9 1/20 0.33
CDK2 P24941 2/20 0.33
EGFR P00533 1/20 0.33
MUSK O15146 1/20 0.33
NTRK1 P04629 1/20 0.33
PRKCB P05771 1/20 0.33
ROS1 P08922 1/20 0.33
PDGFRA P16234 1/20 0.33
FER P16591 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650536 0.90 JAK2 (0.34) SYKJAK2BRD4CDK9CDK1
SCHEMBL22650578 0.85 IKBKB (0.35) JAK2BRD4CDK9CDK1CCNB1
SCHEMBL22650627 0.81 CDK4 (0.39) CDK9CDK1CDK4CCNB1CCND1
SCHEMBL22650620 0.79 CDK2 (0.36) SYKJAK2BRD4CDK9CDK1
SCHEMBL22650630 0.79 CDK9 (0.35) JAK2BRD4CDK9CDK1CCNB1
SCHEMBL22650781 0.75 IKBKB (0.39) SYKJAK2CDK1CDK4CCNB1
SCHEMBL22650514 0.75 CDK4 (0.38) CDK9CDK1CDK4CCNB1CCND1
SCHEMBL22650626 0.74 CDK2 (0.39) SYKJAK2CDK9CDK1CCNB1
SCHEMBL22650549 0.73 ZAP70 (0.42) CDK9CDK1CCNB1IKBKBCHUK
SCHEMBL22650419 0.73 JAK2 (0.38) JAK2BRD4CDK9CDK1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed