SCHEMBL22650561

SCHEMBL22650561

Nc1ccc(N2CCC(NC3CC(F)(F)C3)CC2=O)cn1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.31
FLT3 P36888 1/20 0.31
GCKR Q14397 1/20 0.31
CHRNB2 P17787 1/20 0.30
CHRNA4 P43681 1/20 0.30
AKR1C3 P42330 1/20 0.30
CNR1 P21554 1/20 0.30
LMNA P02545 1/20 0.30
SSTR5 P35346 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650820 0.79 CHRNB2 (0.34) CHRNB2CHRNA4AKR1C3
SCHEMBL22650730 0.73 ALOX5AP (0.40) GCKRCHRNB2CHRNA4AKR1C3
SCHEMBL22650819 0.73 HRH3 (0.39) CHRNB2CHRNA4AKR1C3
SCHEMBL22650822 0.72 CHRNB2 (0.37) GCKRCHRNB2CHRNA4AKR1C3
SCHEMBL18291712 0.72 CKS1B (0.45) CNR1
SCHEMBL22650368 0.70 ALOX5AP (0.37) GCKRCHRNB2CHRNA4AKR1C3
SCHEMBL29462389 0.70 ALOX5AP (0.37) GCKRCHRNB2CHRNA4AKR1C3
SCHEMBL22650818 0.70 PIK3CA (0.37)
SCHEMBL22650562 0.68 PIK3CA (0.35) CHRNB2CHRNA4AKR1C3
SCHEMBL22650566 0.67 DPP4 (0.33) GCKRCHRNB2CHRNA4AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed