SCHEMBL22650566

SCHEMBL22650566

CN(CCF)C1CCN(c2ccc(N)nc2)C(=O)C1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.33
AKR1C3 P42330 1/20 0.32
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31
PIK3CA P42336 3/20 0.31
MTOR P42345 3/20 0.31
TSHR P16473 1/20 0.30
CPB1 P15086 1/20 0.30
BPTF Q12830 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30
GCK P35557 1/20 0.30
GCKR Q14397 1/20 0.30
CHRNB2 P17787 1/20 0.30
CHRNA4 P43681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650910 0.90 DRD3 (0.35) AKR1C3PIK3CAMTOR
SCHEMBL22650368 0.84 ALOX5AP (0.37) AKR1C3ALOX5APFEN1DDB1CRBN
SCHEMBL29462389 0.84 ALOX5AP (0.37) AKR1C3ALOX5APFEN1DDB1CRBN
SCHEMBL22650562 0.81 PIK3CA (0.35) AKR1C3PIK3CAMTORCPB1CHRNB2
SCHEMBL22650573 0.81 LIPE (0.35) DPP4ALOX5APFEN1GCKGCKR
SCHEMBL22650412 0.75 SPR (0.38) PIK3CA
SCHEMBL29491165 0.75 SPR (0.38) PIK3CA
SCHEMBL22650571 0.72 CCR5 (0.39)
SCHEMBL22650730 0.72 ALOX5AP (0.40) AKR1C3ALOX5APFEN1PIK3CAMTOR
SCHEMBL13768888 0.70 CDK4 (0.46) PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed