SCHEMBL22650598

SCHEMBL22650598

CN(C)C1CCN(c2ccc(Nc3nccc(-c4ccn5ncc(C(C)(C)C)c5c4)n3)c(F)c2)C(=O)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.37
JAK2 O60674 2/20 0.35
BRD4 O60885 2/20 0.35
JAK1 P23458 1/20 0.35
BRD2 P25440 1/20 0.35
JAK3 P52333 1/20 0.35
BRD3 Q15059 1/20 0.35
BRDT Q58F21 1/20 0.35
CCNA2 P20248 6/20 0.34
CDK2 P24941 6/20 0.34
CCNA1 P78396 6/20 0.34
ABL1 P00519 4/20 0.34
LYN P07948 3/20 0.34
BCR P11274 2/20 0.34
RIPK2 O43353 1/20 0.34
LCK P06239 1/20 0.34
FYN P06241 1/20 0.34
RET P07949 1/20 0.34
PDGFRB P09619 1/20 0.34
ARAF P10398 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650597 0.89 EGFR (0.37) EGFRJAK2BRD4JAK1BRD2
SCHEMBL22650522 0.84 F10 (0.37) EGFRCCNA2CDK2CCNA1CDK4
SCHEMBL22650428 0.83 CDK4 (0.35) EGFRBRD4CCNA2CDK2CCNA1
SCHEMBL22650421 0.78 JAK2 (0.38) EGFRJAK2BRD4JAK1JAK3
SCHEMBL22650433 0.77 EGFR (0.36) EGFRCDK4CCND3GSK3B
SCHEMBL22650901 0.77 CDK4 (0.45) CCNA2CDK2CCNA1CDK4CCND3
SCHEMBL22650823 0.77 CDK4 (0.45) CCNA2CDK2CCNA1CDK4CCND3
SCHEMBL22650370 0.76 CDK4 (0.35) CCNA2CDK2CCNA1CDK4CCND3
SCHEMBL22650541 0.75 EGFR (0.36) EGFRCCNA2CDK2CCNA1CDK4
SCHEMBL22650922 0.73 F10 (0.38) EGFRJAK2JAK1JAK3MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed