SCHEMBL22650496

SCHEMBL22650496

COc1nc(-c2ccnc(Nc3ccc(N4CCNCC4=O)cc3F)n2)cc2c1ncn2C(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.38
CDK6 Q00534 6/20 0.36
CDK4 P11802 5/20 0.36
F10 P00742 1/20 0.35
ALK Q9UM73 3/20 0.34
CCND1 P24385 2/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
CSF1R P07333 1/20 0.33
CDK1 P06493 3/20 0.32
CCNA2 P20248 2/20 0.32
CCND3 P30281 2/20 0.32
ROS1 P08922 1/20 0.32
MAP4K1 Q92918 1/20 0.32
CCNB1 P14635 2/20 0.32
CDK2 P24941 1/20 0.32
CCNA1 P78396 1/20 0.32
PLK1 P53350 1/20 0.31
PRKD3 O94806 1/20 0.31
PRKCG P05129 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650464 0.89 CDK6 (0.44) EGFRCDK6CDK4F10ALK
SCHEMBL22650501 0.87 CDK2 (0.40) EGFRCDK4CCND1CDK1CCNA2
SCHEMBL22650549 0.83 ZAP70 (0.42) EGFRCDK1CCNA2MAP4K1CCNB1
SCHEMBL22650579 0.79 CDK4 (0.48) CDK6CDK4CCND1CDK1CCNA2
SCHEMBL22650502 0.77 CDK4 (0.43) CDK6CDK4CCND1CSF1RCDK1
SCHEMBL22650624 0.76 EGFR (0.34) EGFRCDK6CCND3
SCHEMBL22650541 0.76 EGFR (0.36) EGFRCDK4ALKCCND1MKNK1
SCHEMBL22650532 0.74 EGFR (0.36) EGFRCDK6CDK4CCND1MKNK1
SCHEMBL22650524 0.74 CDK6 (0.38) EGFRCDK6CDK4F10CCND1
SCHEMBL22650775 0.73 CDK4 (0.44) CDK6CDK4CSF1RCDK1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed