SCHEMBL22650832

SCHEMBL22650832

CNC(=N)Nc1ccc(N2CC(N)CC2=O)cn1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
CDK4 P11802 9/20 0.37
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
CDK1 P06493 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650833 0.84 TSHR (0.36) TSHRMAPK1CDK4CDK1
SCHEMBL22650900 0.78 USP30 (0.34) CDK4CDK1
SCHEMBL22650899 0.78 USP30 (0.34) CDK4CDK1
SCHEMBL22650505 0.74 F10 (0.38) CDK4
SCHEMBL22650606 0.72 WNT3A (0.39) CDK4
SCHEMBL22650942 0.70 CDK4 (0.34) CDK4CDK1
SCHEMBL21580294 0.69 DPP4 (0.54) CYP3A4CYP2C19
SCHEMBL24483273 0.68 CHRNB2 (0.49) CDK4CDK1
SCHEMBL20901706 0.66 TSHR (0.55) TSHRMAPK1LMNAKMT2AMEN1
SCHEMBL20901666 0.66 TSHR (0.55) TSHRMAPK1LMNAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed