SCHEMBL22650900

SCHEMBL22650900

CNC(=N)Nc1ccc(N2CC[C@@H](N(C)C)CC2=O)cn1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.34
CDK4 P11802 18/20 0.33
CCND1 P24385 1/20 0.33
CDK2 P24941 1/20 0.33
CDK1 P06493 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650899 1.00 USP30 (0.34) USP30CDK4CCND1CDK2CDK1
SCHEMBL22650833 0.89 TSHR (0.36) CDK4CDK1
SCHEMBL22650832 0.78 TSHR (0.38) CDK4CDK1
SCHEMBL29462389 0.77 ALOX5AP (0.37)
SCHEMBL22650368 0.77 ALOX5AP (0.37)
SCHEMBL22650505 0.75 F10 (0.38) CDK4CCND1
SCHEMBL22650606 0.73 WNT3A (0.39) CDK4CCND1CDK2
SCHEMBL22650942 0.72 CDK4 (0.34) CDK4CCND1CDK2CDK1
SCHEMBL22650565 0.70 DDB1 (0.38)
SCHEMBL24483273 0.67 CHRNB2 (0.49) CDK4CCND1CDK2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed