SCHEMBL22650833

SCHEMBL22650833

CNC(=N)Nc1ccc(N2CC(N(C)C)CC2=O)cn1

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
CDK4 P11802 17/20 0.36
CDK1 P06493 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650900 0.89 USP30 (0.34) CDK4CDK1
SCHEMBL22650899 0.89 USP30 (0.34) CDK4CDK1
SCHEMBL22650832 0.84 TSHR (0.38) TSHRMAPK1CDK4CDK1
SCHEMBL22650505 0.72 F10 (0.38) CDK4
SCHEMBL22650606 0.70 WNT3A (0.39) CDK4
SCHEMBL22650942 0.69 CDK4 (0.34) CDK4CDK1
SCHEMBL24483273 0.66 CHRNB2 (0.49) CDK4CDK1
SCHEMBL24483448 0.65 WNT3A (0.50) CDK4CDK1
SCHEMBL24483274 0.64 WNT3A (0.57) TSHR
SCHEMBL22650368 0.64 ALOX5AP (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed