SCHEMBL2270596

SCHEMBL2270596

O=C(Nc1cc(-c2ccccc2)ccc1C(=O)O)c1ccc(Cl)cc1Cl

nearest known ligand 0.70

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACLY P53396 8/20 0.70
GRIK1 P39086 3/20 0.62
SERPINE1 P05121 2/20 0.60
PPARG P37231 2/20 0.60
PPARA Q07869 2/20 0.60
SUCNR1 Q9BXA5 1/20 0.60
KDM4E B2RXH2 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
RXFP1 Q9HBX9 1/20 0.59
FLT1 P17948 1/20 0.57
FLT4 P35916 1/20 0.57
KDR P35968 1/20 0.57
HDAC8 Q9BY41 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7038130 0.91 SERPINE1 (0.70) ACLYGRIK1SERPINE1PPARGPPARA
SCHEMBL2269604 0.89 ACLY (0.69) ACLYGRIK1SUCNR1HDAC8HDAC6
SCHEMBL7040843 0.88 PPARG (0.69) ACLYSERPINE1PPARGPPARASUCNR1
SCHEMBL1317521 0.88 ACLY (0.68) ACLYGRIK1SERPINE1SUCNR1
SCHEMBL1308769 0.87 PPARG (0.69) GRIK1PPARGPPARAKDM4ENPSR1
SCHEMBL1315890 0.87 ACLY (0.67) ACLYGRIK1SERPINE1SUCNR1
SCHEMBL2891026 0.86 PPARG (0.68) GRIK1PPARGPPARASUCNR1KDM4E
SCHEMBL2274998 0.85 ACLY (0.80) ACLYGRIK1SERPINE1SUCNR1KDM4E
SCHEMBL14075267 0.83 SERPINE1 (0.80) ACLYGRIK1SERPINE1SUCNR1KDM4E
SCHEMBL2272049 0.83 ACLY (0.78) ACLYGRIK1SERPINE1SUCNR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7999132-B2 Anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO., LTD. (JP) 2011-08-16 US disclosed
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-09-24 US disclosed
EP-1820795-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2007-08-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF MMP13, MMP26, MMP11 ACLY 653/4885GRIK1 2029/4885SERPINE1 101/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.