SCHEMBL2271920

SCHEMBL2271920

O=C(Nc1cc(Oc2cccc(O)c2)ccc1C(=O)O)c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 1/20 0.57
HPSE Q9Y251 1/20 0.56
PYGM P11217 3/20 0.56
PYGL P06737 2/20 0.56
MEN1 O00255 2/20 0.56
PKM P14618 2/20 0.56
KMT2A Q03164 2/20 0.56
TDP1 Q9NUW8 2/20 0.55
MAPT P10636 2/20 0.55
GRIK1 P39086 1/20 0.55
AKR1C4 P17516 3/20 0.54
AKR1C3 P42330 3/20 0.54
AKR1C2 P52895 3/20 0.54
AKR1C1 Q04828 3/20 0.54
GALK1 P51570 1/20 0.54
CASP6 P55212 1/20 0.54
MCL1 Q07820 1/20 0.54
PLEC Q15149 1/20 0.54
NR1H4 Q96RI1 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2275060 0.94 AKR1C4 (0.59) SERPINE1PYGMPYGLMEN1PKM
SCHEMBL2271588 0.91 SERPINE1 (0.64) SERPINE1HPSEPYGMPYGLMEN1
SCHEMBL2274898 0.90 SERPINE1 (0.60) SERPINE1HPSEPYGMPYGLMEN1
SCHEMBL2276745 0.88 SERPINE1 (0.65) SERPINE1HPSEPYGMPYGLMEN1
SCHEMBL2272040 0.86 PGR (0.69) HPSEPYGMPYGLMEN1PKM
SCHEMBL2269555 0.86 HPSE (0.55) SERPINE1HPSEPYGMPYGLMEN1
SCHEMBL2273166 0.86 GFER (0.61) SERPINE1HPSEPYGMPYGLMEN1
SCHEMBL2274838 0.86 SERPINE1 (0.66) SERPINE1HPSEPYGMPYGLMEN1
SCHEMBL2275544 0.84 FABP1 (0.61) SERPINE1PYGMMEN1PKMKMT2A
SCHEMBL2273044 0.83 CYP2C9 (0.61) SERPINE1PYGMPYGLMEN1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101094829-B novel anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO.,LTD. (JP) 2012-02-08 CN disclosed
US-7999132-B2 Anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO., LTD. (JP) 2011-08-16 US disclosed
US-7999132-B2 Anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO., LTD. (JP) 2011-08-16 US disclosed
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-09-24 US disclosed
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-09-24 US disclosed
CN-101094829-A Novel anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO LTD (JP) 2007-12-26 CN disclosed
EP-1820795-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2007-08-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF MMP13, MMP26, MMP11 SERPINE1 101/4885HPSE 1324/4885PYGM 1299/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.